SCHEMBL5314528

SCHEMBL5314528

O=C(Nc1cc(C(=O)Nc2ccccc2O)cc(C(=O)Nc2ccccc2O)c1)c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.59
KMT2A Q03164 4/20 0.59
MEN1 O00255 3/20 0.59
RAB9A P51151 3/20 0.59
TP53 P04637 3/20 0.59
KCNMA1 Q12791 2/20 0.56
HDAC1 Q13547 1/20 0.56
HDAC2 Q92769 1/20 0.56
PKM P14618 2/20 0.56
TOP1 P11387 1/20 0.56
TOP2A P11388 1/20 0.56
TOP2B Q02880 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
KCNK3 O14649 2/20 0.54
KCNK9 Q9NPC2 2/20 0.54
FKBP5 Q13451 1/20 0.54
GAA P10253 2/20 0.53
LMNA P02545 1/20 0.53
HTT P42858 1/20 0.53
MDM4 O15151 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17200812 0.93 NPC1 (0.52) NPC1KMT2AMEN1RAB9ATP53
SCHEMBL1470784 0.88 NPC1 (0.73) NPC1KMT2AMEN1RAB9ATP53
SCHEMBL4946074 0.88 NPC1 (0.73) NPC1KMT2AMEN1RAB9ATP53
SCHEMBL19630945 0.87 HDAC1 (0.66) NPC1KMT2AMEN1RAB9ATP53
SCHEMBL462324 0.84 MEN1 (0.66) NPC1KMT2AMEN1RAB9ATP53
SCHEMBL2332797 0.83 KMT2A (0.77) KMT2AMEN1RAB9APKML3MBTL1
SCHEMBL6029925 0.82 NPC1 (0.82) NPC1KMT2AMEN1RAB9ATP53
SCHEMBL3860173 0.80 TOP1 (0.59) NPC1KMT2AMEN1RAB9ATP53
SCHEMBL7817331 0.80 HDAC1 (0.69) NPC1KMT2AMEN1RAB9AKCNMA1
SCHEMBL3864321 0.80 TOP1 (0.62) NPC1KMT2AMEN1RAB9ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070148185-A1 Novel therapeutic target for protozoal diseases VIRGINIA POLYTECHNIC INSTITUTE AND STATE UNIVERSITY 2007-06-28 US claimed
WO-2007047579-A2 A NOVEL THERAPEUTIC TARGET FOR PROTOZOAL DISEASES VIRGINIA TECH INTELLECTUAL PROPERTIES, INC. (US) 2007-04-26 WO claimed
EP-2931280-B1 METHODS AND COMPOSITIONS FOR INHIBITING CNKSR1 PHUSIS THERAPEUTICS INC (US) 2018-02-14 EP disclosed