SCHEMBL5314786

SCHEMBL5314786

CNC1CN(C)CCn2c1nc(C(=O)O)c(O)c2=O

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ERCC1 P07992 2/20 0.35
ERCC4 Q92889 2/20 0.35
FEN1 P39748 1/20 0.35
KCNH2 Q12809 1/20 0.30
CYP2C9 P11712 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2206687 0.88 NPSR1 (0.32) ERCC1ERCC4FEN1
SCHEMBL2208054 0.66 KCNH2 (0.58) ERCC1ERCC4FEN1KCNH2CYP2C9
SCHEMBL5757341 0.66 CYP2C9 (0.38) ERCC1ERCC4FEN1KCNH2CYP2C9
SCHEMBL2202249 0.65 ALDH1A1 (0.43) ERCC1ERCC4FEN1KCNH2CYP2C9
SCHEMBL12529315 0.60 ALDH1A1 (0.36) KCNH2
SCHEMBL13672437 0.60 NPSR1 (0.36) ERCC1ERCC4FEN1
SCHEMBL12471410 0.59 ERCC1 (0.54) ERCC1ERCC4FEN1
SCHEMBL5528388 0.58 ERCC1 (0.33) ERCC1ERCC4FEN1
SCHEMBL5336044 0.58 MAPT (0.37) ERCC1ERCC4FEN1
SCHEMBL13815129 0.57 F10 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1866313-A1 HIV INTEGRASE INHIBITORS Istituto di Richerche di Biologia Molecolare P. Angeletti S.p.A. (IT) 2007-12-19 EP disclosed
WO-2006103399-A1 HIV INTEGRASE INHIBITORS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P ANGELETTI SPA (IT) 2006-10-05 WO disclosed