SCHEMBL5314947

SCHEMBL5314947

N=C(NO)c1nccc2nc(C(F)(F)F)ccc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 5/20 0.37
CNR2 P34972 3/20 0.36
NT5E P21589 1/20 0.34
TAS2R14 Q9NYV8 1/20 0.34
CLK4 Q9HAZ1 3/20 0.34
ACVR1 Q04771 3/20 0.34
GSK3A P49840 3/20 0.33
GSK3B P49841 3/20 0.33
IGF1R P08069 1/20 0.33
PRKD3 O94806 1/20 0.33
MAP4K4 O95819 1/20 0.33
MARK3 P27448 1/20 0.33
KDR P35968 1/20 0.33
MAPKAPK2 P49137 1/20 0.33
PRKCZ Q05513 1/20 0.33
PRKAA1 Q13131 1/20 0.33
PAK1 Q13153 1/20 0.33
STK3 Q13188 1/20 0.33
TAOK1 Q7L7X3 1/20 0.33
HIPK4 Q8NE63 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5261941 0.84 CNR2 (0.36) CNR2NT5ETAS2R14CLK4ACVR1
SCHEMBL13853244 0.80 TAS2R14 (0.42) HDAC4CNR2TAS2R14CLK4ACVR1
SCHEMBL13853248 0.79 CNR2 (0.35) CNR2NT5ETAS2R14CLK4ACVR1
SCHEMBL13853240 0.75 PDPK1 (0.35) CNR2NT5ETAS2R14CLK4ACVR1
SCHEMBL5314951 0.75 PDPK1 (0.35) CNR2NT5ETAS2R14CLK4ACVR1
SCHEMBL17610 0.73 HDAC4 (0.38) HDAC4TAS2R14SYK
SCHEMBL13853234 0.71 CYP2A6 (0.40) NT5E
SCHEMBL5265938 0.71 NOS3 (0.40) NT5ECLK4ACVR1GSK3AGSK3B
SCHEMBL4187576 0.71 NT5E (0.42) NT5ETAS2R14CLK4ACVR1GSK3A
SCHEMBL5264358 0.71 MAPT (0.46) NT5ETAS2R14CLK4ACVR1GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1824828-A2 PYRIDINE BASED COMPOUNDS USEFUL AS INTERMEDIATES FOR PHARMACEUTICAL OR AGRICULTURAL END-PRODUCTS Peakdale Molecular Limited (GB) 2007-08-29 EP disclosed
WO-2006059103-A2 PYRIDINE BASED COMPOUNDS USEFUL AS INTERMEDIATES FOR PHARMACEUTICAL OR AGRICULTURAL END-PRODUCTS PEAKDALE MOLECULAR LIMITED (GB) 2006-06-08 WO disclosed