SCHEMBL5314951

SCHEMBL5314951

NC(=NO)c1nccc2nc(C(F)(F)F)ccc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.35
NPSR1 Q6W5P4 1/20 0.34
CNR2 P34972 2/20 0.33
SYK P43405 3/20 0.32
KMT2A Q03164 1/20 0.32
CLK4 Q9HAZ1 3/20 0.31
ACVR1 Q04771 2/20 0.31
NPC1 O15118 1/20 0.31
GAA P10253 1/20 0.31
RAB9A P51151 1/20 0.31
TAS2R14 Q9NYV8 1/20 0.31
ADORA2A P29274 1/20 0.31
ADORA1 P30542 1/20 0.31
GSK3A P49840 2/20 0.31
GSK3B P49841 2/20 0.31
IGF1R P08069 1/20 0.31
PRKD3 O94806 1/20 0.31
MAP4K4 O95819 1/20 0.31
MARK3 P27448 1/20 0.31
KDR P35968 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13853240 1.00 PDPK1 (0.35) PDPK1NPSR1CNR2SYKKMT2A
SCHEMBL13853248 0.84 CNR2 (0.35) CNR2SYKCLK4ACVR1TAS2R14
SCHEMBL5261941 0.82 CNR2 (0.36) CNR2SYKCLK4ACVR1TAS2R14
SCHEMBL13853244 0.79 TAS2R14 (0.42) CNR2SYKCLK4ACVR1TAS2R14
SCHEMBL5314947 0.75 HDAC4 (0.37) CNR2SYKCLK4ACVR1TAS2R14
SCHEMBL5265938 0.73 NOS3 (0.40) SYKKMT2ACLK4ACVR1GSK3A
SCHEMBL17608 0.72 ADRB1 (0.36) PDPK1NPSR1SYKKMT2ANPC1
SCHEMBL17609 0.72 ADRB1 (0.36) PDPK1NPSR1SYKKMT2ANPC1
SCHEMBL13853234 0.70 CYP2A6 (0.40) KMT2ANT5EMAPT
SCHEMBL4187576 0.70 NT5E (0.42) SYKCLK4ACVR1TAS2R14ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1824828-A2 PYRIDINE BASED COMPOUNDS USEFUL AS INTERMEDIATES FOR PHARMACEUTICAL OR AGRICULTURAL END-PRODUCTS Peakdale Molecular Limited (GB) 2007-08-29 EP disclosed
WO-2006059103-A2 PYRIDINE BASED COMPOUNDS USEFUL AS INTERMEDIATES FOR PHARMACEUTICAL OR AGRICULTURAL END-PRODUCTS PEAKDALE MOLECULAR LIMITED (GB) 2006-06-08 WO disclosed