SCHEMBL5317370

SCHEMBL5317370

O=C(C=CN1CCC(C(CO)N2CCC(c3c[nH]c4c3ccc[n+]4[O-])CC2)CC1)c1cc(F)cc(F)c1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 20/20 0.55
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C19 P33261 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5946893 0.83 CCR2 (0.76) CCR2CYP3A4CYP2D6CYP2C19
SCHEMBL5318246 0.78 CCR2 (0.70) CCR2
SCHEMBL5320143 0.77 CCR2 (0.71) CCR2CYP3A4CYP2D6CYP2C19
SCHEMBL5315276 0.75 CCR2 (0.44) CCR2CYP3A4CYP2D6CYP2C19
SCHEMBL5346961 0.75 CCR2 (0.54) CCR2
SCHEMBL5351353 0.73 KMT2A (0.52) CCR2
SCHEMBL5946910 0.71 CCR2 (1.00) CCR2CYP3A4CYP2D6CYP2C19
SCHEMBL5946913 0.71 CCR2 (1.00) CCR2CYP3A4CYP2D6CYP2C19
SCHEMBL5357090 0.70 CCR2 (0.53) CCR2CYP3A4CYP2D6CYP2C19
SCHEMBL5328493 0.68 CCR2 (0.54) CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1802602-A1 SUBSTITUTED DIPIPERDINE CCR2 ANTAGONISTS JANSSEN PHARMACEUTICA N.V. (BE) 2007-07-04 EP disclosed
WO-2006036527-A1 SUBSTITUTED DIPIPERDINE CCR2 ANTAGONISTS JANSSEN PHARMACEUTICA, N.V. (BE) 2006-04-06 WO disclosed