SCHEMBL5317628

SCHEMBL5317628

CN(Cc1ccc(C#N)cc1)C(=O)CN1CC2CN(CCc3c(F)cccc3F)CC(C1)O2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 2/20 0.41
CCR5 P51681 2/20 0.37
PLA2G7 Q13093 1/20 0.37
KCNH2 Q12809 4/20 0.36
AGTR2 P50052 1/20 0.36
CCR1 P32246 1/20 0.35
TACR3 P29371 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
CCR3 P51677 1/20 0.34
CHRM2 P08172 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
HCRTR1 O43613 1/20 0.34
HCRTR2 O43614 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KCNJ1 P48048 2/20 0.34
GRIN1 Q05586 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5319745 0.87 KMT2A (0.43) CCR5KCNH2AGTR2MEN1KMT2A
SCHEMBL5314383 0.83 CCR1 (0.39) NSD2CCR5PLA2G7KCNH2AGTR2
SCHEMBL5314580 0.82 CCR5 (0.39) NSD2CCR5PLA2G7AGTR2MEN1
SCHEMBL5320812 0.80 NSD2 (0.42) NSD2CCR5AGTR2CCR1MEN1
SCHEMBL5317011 0.78 KCNH2 (0.47) KCNH2MEN1SMN1; SMN2GRIN1GRIN2B
SCHEMBL3127996 0.73 KCNH2 (0.54) KCNH2
SCHEMBL2967576 0.72 KCNH2 (0.47) KCNH2KCNJ1
SCHEMBL3117605 0.72 KCNH2 (0.52) KCNH2KMT2ACCR3
SCHEMBL5317641 0.69 MEN1 (0.42) NSD2CCR5KCNH2MEN1KMT2A
SCHEMBL5317453 0.69 KMT2A (0.48) KCNH2KMT2AALDH1A1POLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007069986-A1 NEW OXABISPIDINE COMPOUNDS FOR THE TREATMENT OF CARDIAC ARRHYTHMIAS ASTRAZENECA AB (SE) 2007-06-21 WO claimed