SCHEMBL5314580

SCHEMBL5314580

CN(Cc1ccc(C#N)cc1)C(=O)CN1CC2CN(CCc3ccccc3C(F)(F)F)CC(C1)O2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 2/20 0.39
POLB P06746 2/20 0.38
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
NSD2 O96028 1/20 0.37
KDM4E B2RXH2 5/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
ATM Q13315 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
PGR P06401 2/20 0.36
GAA P10253 2/20 0.36
MAPK1 P28482 1/20 0.36
ALDH1A1 P00352 4/20 0.36
AGTR2 P50052 1/20 0.36
PLA2G7 Q13093 1/20 0.35
MAPT P10636 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5314383 0.87 CCR1 (0.39) CCR5POLBNSD2MEN1KMT2A
SCHEMBL5319745 0.85 KMT2A (0.43) CCR5POLBMEN1KMT2AALDH1A1
SCHEMBL5316681 0.83 POLB (0.40) POLBKDM4EALDH1A1HTT
SCHEMBL5317628 0.82 NSD2 (0.41) CCR5POLBNSD2MEN1KMT2A
SCHEMBL5320812 0.77 NSD2 (0.42) CCR5POLBSLC6A2SLC6A4NSD2
SCHEMBL5317011 0.77 KCNH2 (0.47) MEN1
SCHEMBL5316954 0.72 POLB (0.44) POLBKDM4EMEN1KMT2AALDH1A1
SCHEMBL2967576 0.71 KCNH2 (0.47)
SCHEMBL5315901 0.70 DRD2 (0.49) POLBKDM4EMEN1KMT2AGAA
SCHEMBL5317641 0.69 MEN1 (0.42) CCR5NSD2MEN1KMT2AOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007069986-A1 NEW OXABISPIDINE COMPOUNDS FOR THE TREATMENT OF CARDIAC ARRHYTHMIAS ASTRAZENECA AB (SE) 2007-06-21 WO claimed