SCHEMBL5319227

SCHEMBL5319227

CCCS(=O)(=O)c1ccc(CN2CCC(c3c(F)cc(F)c(NC(=O)C(C)C)c3F)CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 9/20 0.44
ADRA1A P35348 4/20 0.44
ALDH1A1 P00352 1/20 0.41
MAPK1 P28482 1/20 0.41
KCNH2 Q12809 1/20 0.36
GPR119 Q8TDV5 1/20 0.36
RORC P51449 1/20 0.35
ACKR3 P25106 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5319226 0.89 DRD2 (0.46) DRD2ADRA1AKCNH2GPR119ACKR3
SCHEMBL4637063 0.81 DRD2 (0.49) DRD2ADRA1A
SCHEMBL4617156 0.81 DRD2 (0.50) DRD2ADRA1A
SCHEMBL5347220 0.80 DRD2 (0.52) DRD2ADRA1AALDH1A1MAPK1
SCHEMBL5324228 0.77 DRD2 (0.63) DRD2ADRA1AALDH1A1MAPK1
SCHEMBL5322079 0.71 DRD2 (0.49) DRD2ADRA1AKCNH2GPR119
SCHEMBL5321967 0.71 GAA (0.41) DRD2ALDH1A1KCNH2RORC
SCHEMBL5319269 0.71 MCHR1 (0.56) DRD2ADRA1AKCNH2
SCHEMBL6000445 0.70 UBE2M (0.39)
SCHEMBL4765040 0.69 KDM4E (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007114902-A2 ALKYLTHIOBENZYLPIPERIDINE COMPOUNDS H.LUNDBECK A/S (DK) 2007-10-11 WO claimed