SCHEMBL5320139

SCHEMBL5320139

COC(=O)c1ccccc1-c1ccccc1C(c1ccc(NC2=NCCN2)cc1)N1N=C(C2CCCCC2)c2ccccc2NC1=O

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTH1R Q03431 2/20 0.43
PTGIR P43119 8/20 0.34
ADRA2A P08913 5/20 0.33
ADRA2B P18089 5/20 0.33
ADRA2C P18825 5/20 0.33
ADRA1D P25100 1/20 0.32
ADRA1A P35348 1/20 0.32
ADRA1B P35368 1/20 0.32
PDE4D Q08499 1/20 0.31
PDE7A Q13946 1/20 0.31
ITGB3 P05106 1/20 0.31
ITGAV P06756 1/20 0.31
ITGA2B P08514 1/20 0.31
CCKBR P32239 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5320137 0.73 PTH1R (0.72) PTH1RCCKBR
SCHEMBL5321430 0.67 CYP19A1 (0.36) PTH1RCCKBR
SCHEMBL5320787 0.61 PTH1R (1.00) PTH1RPTGIRCCKBR
SCHEMBL6829822 0.60 CCKBR (0.40) PTH1RCCKBR
SCHEMBL14566393 0.60 PTH1R (0.79) PTH1R
SCHEMBL5494976 0.59 PTH1R (0.84) PTH1RPTGIRADRA2AADRA2BADRA2C
SCHEMBL5281350 0.59 PTH1R (0.38) PTH1RPDE4DCCKBR
SCHEMBL5287497 0.59 PTH1R (0.50) PTH1RPDE4D
SCHEMBL3909395 0.58 PDE4A (0.45) PDE4DCCKBR
SCHEMBL9178572 0.58 NISCH (0.46) PTH1RADRA2AADRA2BADRA2CADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129120-A9 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2007-03-22 WO disclosed
WO-2006129120-A2 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2006-12-07 WO disclosed