SCHEMBL5320835

SCHEMBL5320835

COc1ccc(N2CCN(C)CC2)c2nc(C(=O)O)cc(O)c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
HPGD P15428 2/20 0.47
TSHR P16473 2/20 0.47
CASP1 P29466 1/20 0.47
CASP7 P55210 1/20 0.47
GFER P55789 1/20 0.42
HSD17B10 Q99714 1/20 0.42
GPR35 Q9HC97 1/20 0.42
HTR1B P28222 6/20 0.41
HTR1A P08908 5/20 0.41
HTR1D P28221 5/20 0.41
DRD2 P14416 1/20 0.40
DRD3 P35462 1/20 0.40
HTR6 P50406 3/20 0.40
HTR2A P28223 2/20 0.40
HTR2C P28335 2/20 0.40
HTR7 P34969 1/20 0.40
ALOX15 P16050 1/20 0.40
ERAP1 Q9NZ08 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5319256 0.85 KDM4A (0.42) KDM4EALDH1A1HSD17B10DRD2DRD3
Hydrochloric Acid SCHEMBL6080168 0.75 HTR6 (0.45) KDM4EALDH1A1HTR1BHTR1AHTR1D
SCHEMBL4991445 0.74 HTR1B (0.63) KDM4EALDH1A1HPGDTSHRCASP1
Hydrochloric Acid SCHEMBL4990186 0.73 HTR1B (0.62) KDM4EALDH1A1HPGDTSHRCASP1
SCHEMBL6591671 0.71 KDM4A (0.48) KDM4EALDH1A1HTR6MEN1USP2
SCHEMBL6592438 0.71 GPR35 (0.51) KDM4EALDH1A1HPGDTSHRHSD17B10
Hydrochloric Acid SCHEMBL6079508 0.71 KDM4A (0.47) KDM4EALDH1A1HTR6MEN1USP2
SCHEMBL6597066 0.70 GPR35 (0.47) KDM4EALDH1A1HPGDGPR35ALOX15
SCHEMBL6601321 0.70 GPR35 (0.44) KDM4EALDH1A1HPGDTSHRGPR35
SCHEMBL5827458 0.70 HTR1D (0.55) HTR1BHTR1AHTR1DDRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007097697-A1 THERAPEUTIC QUINOLINE COMPOUNDS THAT ARE 5HT1B MODULATORS ASTRAZENECA AB (SE) 2007-08-30 WO disclosed