SCHEMBL5322121

SCHEMBL5322121

CS(=O)(=O)OCCc1ccc(S(=O)(=O)c2ccc(F)c(F)c2)cc1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA1 P00915 5/20 0.42
CA2 P00918 5/20 0.42
HTR2A P28223 3/20 0.41
HTR2C P28335 2/20 0.41
HTR6 P50406 1/20 0.40
NAMPT P43490 4/20 0.39
KCNH2 Q12809 2/20 0.37
VCAM1 P19320 1/20 0.36
F2 P00734 1/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
TSHR P16473 1/20 0.35
TMPRSS4 Q9NRS4 1/20 0.35
PTGS2 P35354 1/20 0.35
CYP26B1 Q9NR63 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5344844 0.85 DAO (0.40) CA1CA2KCNH2TSHRPTGS2
SCHEMBL3258334 0.78 CA2 (0.50) CA1CA2KCNH2TSHR
SCHEMBL5321788 0.77 CA2 (0.51) CA1CA2HTR2AHTR2CHTR6
SCHEMBL980388 0.76 CA1 (0.44) CA1CA2HTR2AHTR2CKCNH2
SCHEMBL31456176 0.76 VCAM1 (0.55) CA1CA2HTR2AHTR2CHTR6
SCHEMBL14248769 0.75 DAO (0.41) CA1CA2PTGS2
SCHEMBL4318681 0.74 VCAM1 (0.57) CA1CA2HTR6VCAM1TSHR
SCHEMBL30838118 0.74 VCAM1 (0.57) CA1CA2HTR6VCAM1TSHR
SCHEMBL7463569 0.73 PTGS2 (0.45) HTR2AHTR2CHTR6PTGS2
SCHEMBL1284072 0.73 CA1 (0.43) CA1CA2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007114916-A2 ARYLBENZYLPIPERIDINE COMPOUNDS H. LUNDBECK A/S (DK) 2007-10-11 WO disclosed