SCHEMBL5326263

SCHEMBL5326263

C=CCONC1CN(C(=O)O)Nc2ccccc21

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 2/20 0.33
CA1 P00915 2/20 0.32
CA2 P00918 2/20 0.32
THRB P10828 1/20 0.32
CYP3A4 P08684 1/20 0.31
CXCR5 P32302 3/20 0.31
TEAD1 P28347 1/20 0.31
TEAD3 Q99594 1/20 0.31
CHRM1 P11229 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5322672 0.90 CASP1 (0.37) CASP1CA1CA2CYP3A4CHRM1
SCHEMBL5318595 0.83 NPC1 (0.37)
SCHEMBL4862831 0.77 TDP1 (0.34) CASP1CA1CA2
SCHEMBL5253676 0.76 ACE (0.36) CA1CA2CYP3A4CHRM1
SCHEMBL5188020 0.74 CYP19A1 (0.36) CHRM1
SCHEMBL5272076 0.71 CA1 (0.31) CA1CA2
Hydrochloric Acid SCHEMBL4853976 0.70 CA1 (0.31) CA1CA2
SCHEMBL5257111 0.70 TSHR (0.38) CASP1CA1CA2CYP3A4CXCR5
SCHEMBL5255776 0.70 HSD11B1 (0.32)
SCHEMBL4696280 0.67 NPC1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537117-B1 BENZOTRIAZABICYCLIC DERIVATIVES AND USE THEREOF AS BETA-LACTAMASE INHIBITORS AND ANTI-BACTERIAL AGENTS AVENTIS PHARMA SA (FR) 2007-01-17 EP disclosed