SCHEMBL5326522

SCHEMBL5326522

C#CCCCCCCOC(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.52
HRH4 Q9H3N8 1/20 0.44
TK2 O00142 10/20 0.44
TK1 P04183 1/20 0.42
CYP3A4 P08684 3/20 0.38
ALOX15 P16050 2/20 0.38
ALDH1A1 P00352 1/20 0.38
DUT P33316 1/20 0.36
SLC6A1 P30531 1/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
HSD17B10 Q99714 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5323607 0.98 KIF11 (0.53) KIF11HRH4TK2TK1CYP3A4
SCHEMBL5325668 0.93 KIF11 (0.55) KIF11HRH4TK2TK1CYP3A4
SCHEMBL9371526 0.87 KIF11 (0.57) KIF11HRH4TK2TK1CYP3A4
SCHEMBL9637348 0.78 KIF11 (0.55) KIF11HRH4TK2TK1ALOX15
SCHEMBL5820308 0.78 KIF11 (0.55) KIF11HRH4TK2TK1CYP3A4
SCHEMBL25077435 0.78 KIF11 (0.55) KIF11HRH4TK2TK1CYP3A4
SCHEMBL5820348 0.78 KIF11 (0.55) KIF11HRH4TK2TK1CYP3A4
SCHEMBL25077100 0.78 KIF11 (0.55) KIF11HRH4TK2TK1CYP3A4
SCHEMBL21411547 0.78 KIF11 (0.55) KIF11HRH4TK2TK1CYP3A4
SCHEMBL914263 0.78 KIF11 (0.55) KIF11HRH4TK2TK1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0827423-B1 FUNCTIONALIZED CHAIN EXTENDED INITIATORS FOR ANIONIC POLYMERIZATION FMC CORP (US) 2007-12-12 EP claimed
US-4179451-A HYPOTENSIVE, ANTIULCER, BRONCHODILATOR, ANTICONVULSANTS OR ANTIMICROBIAL AGENTS AMERICAN CYANAMID COMPANY (US) 1979-12-18 US disclosed
US-4107441-A HYPOTENSIVE, ANTIULCER, BRONCHODILATORS, ANTIMICROBIAL, ANTICONVULSANTS AMERICAN CYANAMID COMPANY (US) 1978-08-15 US disclosed
US-4061672-A Derivatives of 9-hydroxy-13-trans-prostenoic acid AMERICAN CYANAMID COMPANY (US) 1977-12-06 US disclosed
US-RE29469-E PROSTAGLANDINS; BRONCHODILATORS, HYPOTENSIVES, ANTIULCER AGENTS AMERICAN CYANAMID COMPANY (US) 1977-11-08 US disclosed
US-3950406-A BRONCHODILATORS, HYPOTENSIVE, ANTIULCER AMERICAN CYANAMID COMPANY (US) 1976-04-13 US disclosed