SCHEMBL5328398

SCHEMBL5328398

CC(=O)Oc1cccc(N)c1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.46
PTGS2 P35354 5/20 0.46
KDM4E B2RXH2 4/20 0.46
TDP1 Q9NUW8 3/20 0.46
ALDH1A1 P00352 3/20 0.46
HSD17B10 Q99714 2/20 0.46
BLM P54132 2/20 0.46
ESR1 P03372 1/20 0.46
ITGB3 P05106 1/20 0.46
ITGA2B P08514 1/20 0.46
HMGB1 P09429 1/20 0.46
HPGD P15428 1/20 0.46
TSHR P16473 1/20 0.46
GGT1 P19440 1/20 0.46
PTGS1 P23219 1/20 0.46
NAPRT Q6XQN6 1/20 0.46
ACHE P22303 1/20 0.45
LMNA P02545 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10448816 0.86 KDM4E (0.53) MAPK1PTGS2KDM4ETDP1ALDH1A1
SCHEMBL27966057 0.83 KDM4E (0.42) MAPK1PTGS2KDM4ETDP1ALDH1A1
SCHEMBL3188087 0.82 KDM4E (0.50) MAPK1PTGS2KDM4ETDP1ALDH1A1
SCHEMBL907658 0.81 ACHE (0.61) MAPK1PTGS2KDM4ETDP1ALDH1A1
SCHEMBL6691258 0.81 MAPK1 (0.49) MAPK1PTGS2KDM4ETDP1ALDH1A1
SCHEMBL31612517 0.81 MAPK1 (0.49) MAPK1PTGS2KDM4ETDP1ALDH1A1
SCHEMBL1159881 0.81 ESR1 (0.42) MAPK1KDM4EALDH1A1HSD17B10ESR1
SCHEMBL362353 0.80 PTGS2 (0.57) MAPK1PTGS2KDM4ETDP1ALDH1A1
SCHEMBL4565094 0.80 ALDH1A1 (0.43) MAPK1PTGS2KDM4ETDP1ALDH1A1
SCHEMBL27603303 0.80 TSHR (0.46) MAPK1PTGS2KDM4ETDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007144729-A1 AN IMPROVED PROCESS FOR THE PREPARATION OF CLOPIDOGREL ORCHID CHEMICALS & PHARMACEUTICALS LIMITED (IN) 2007-12-21 WO disclosed