SCHEMBL5328641

SCHEMBL5328641

Cn1ccnc1S(=O)(=O)Nc1ccc(C(=O)O)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
TSHR P16473 2/20 0.47
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47
TDP1 Q9NUW8 2/20 0.45
HTT P42858 1/20 0.45
MCL1 Q07820 1/20 0.44
GAA P10253 2/20 0.44
GFER P55789 1/20 0.44
POLB P06746 3/20 0.44
TP53 P04637 1/20 0.44
CTSL P07711 1/20 0.43
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43
MAPK1 P28482 1/20 0.43
PIK3C3 Q8NEB9 1/20 0.43
IKBKB O14920 1/20 0.42
FABP4 P15090 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8230281 0.72 MCL1 (0.45) CA1CA2MCL1PIK3C3
SCHEMBL1473418 0.70 TRPM5 (0.50) TSHRCA1CA2POLBMEN1
SCHEMBL24051973 0.70 MCL1 (0.46) CA12CA1CA2CA9TDP1
SCHEMBL5330598 0.70 CA12 (0.67) ALDH1A1CA12CA1CA2CA9
SCHEMBL5332392 0.70 TSHR (0.52) ALDH1A1TSHRCA12CA1CA2
SCHEMBL5329438 0.69 ALDH1A1 (0.50) ALDH1A1TSHRCA12CA1CA2
SCHEMBL25072770 0.69 CA12 (0.49) ALDH1A1TSHRCA12CA1CA2
SCHEMBL118340 0.68 KEAP1 (0.59) ALDH1A1CA12CA1CA2CA9
SCHEMBL24051971 0.67 MCL1 (0.44) CA12CA1CA2CA9TDP1
SCHEMBL893905 0.67 CA12 (0.73) ALDH1A1TSHRCA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007144379-A1 BICYCLIC COMPOUNDS USEFUL AS CATHEPSIN S INBHIBITORS MEDIVIR AB (SE) 2007-12-21 WO disclosed
WO-2007144379-A1 BICYCLIC COMPOUNDS USEFUL AS CATHEPSIN S INBHIBITORS MEDIVIR AB (SE) 2007-12-21 WO disclosed