SCHEMBL5329256

SCHEMBL5329256

NNC(=O)CSc1nnc(-c2ccc3c(c2)OCO3)n1C1CCCCC1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.58
LMNA P02545 1/20 0.57
MAPK1 P28482 1/20 0.57
CYP3A4 P08684 1/20 0.56
CYP2D6 P10635 1/20 0.56
TSHR P16473 2/20 0.56
SMN1; SMN2 Q16637 3/20 0.52
GAA P10253 1/20 0.51
KMT2A Q03164 2/20 0.51
HPGD P15428 1/20 0.51
MEN1 O00255 1/20 0.51
MDM2 Q00987 1/20 0.51
ADRB2 P07550 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5329135 0.84 ALDH1A1 (0.65) ALDH1A1LMNAMAPK1CYP3A4CYP2D6
SCHEMBL5329766 0.83 GAA (0.64) ALDH1A1LMNATSHRGAAKMT2A
SCHEMBL5338355 0.82 TSHR (0.59) ALDH1A1CYP3A4CYP2D6TSHRGAA
SCHEMBL5422195 0.82 GAA (0.62) ALDH1A1LMNATSHRGAAKMT2A
SCHEMBL14542393 0.81 MEN1 (0.54) ALDH1A1LMNAMAPK1CYP3A4CYP2D6
SCHEMBL5328964 0.81 SMN1; SMN2 (0.75) ALDH1A1LMNAMAPK1TSHRSMN1; SMN2
SCHEMBL14542019 0.80 MEN1 (0.57) ALDH1A1LMNAMAPK1CYP3A4CYP2D6
SCHEMBL5330985 0.80 TSHR (0.56) ALDH1A1LMNATSHRGAAKMT2A
SCHEMBL5336800 0.78 KMT2A (0.80) ALDH1A1LMNATSHRGAAKMT2A
SCHEMBL5425561 0.77 RXFP1 (0.60) ALDH1A1LMNAMAPK1CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007047394-A2 THIOTRIAZOLYL DERIVATIVES EPIX DELAWARE, INC. (US) 2007-04-26 WO disclosed