SCHEMBL5338355

SCHEMBL5338355

NNC(=O)CSc1nnc(-c2ccc(F)cc2)n1C1CCCCC1

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.59
GAA P10253 3/20 0.59
MEN1 O00255 5/20 0.56
KMT2A Q03164 5/20 0.56
HPGD P15428 2/20 0.56
MDM2 Q00987 1/20 0.56
ADRB2 P07550 1/20 0.54
ALDH1A1 P00352 4/20 0.54
KDM4E B2RXH2 2/20 0.54
RXFP1 Q9HBX9 1/20 0.48
HSD17B10 Q99714 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5329766 0.90 GAA (0.64) TSHRGAAMEN1KMT2AHPGD
SCHEMBL5422195 0.89 GAA (0.62) TSHRGAAMEN1KMT2AHPGD
SCHEMBL5330985 0.87 TSHR (0.56) TSHRGAAMEN1KMT2AHPGD
SCHEMBL5336800 0.82 KMT2A (0.80) TSHRGAAMEN1KMT2AHPGD
SCHEMBL5329256 0.82 ALDH1A1 (0.58) TSHRGAAMEN1KMT2AHPGD
SCHEMBL5332292 0.82 GAA (0.58) TSHRGAAMEN1KMT2AHPGD
SCHEMBL5331047 0.80 KMT2A (0.62) TSHRGAAMEN1KMT2AHPGD
SCHEMBL5330488 0.80 KMT2A (0.62) TSHRGAAMEN1KMT2AHPGD
SCHEMBL5416217 0.79 ALDH1A1 (0.60) TSHRGAAMEN1KMT2AHPGD
SCHEMBL5330577 0.78 TDP1 (0.59) TSHRGAAHPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007047394-A2 THIOTRIAZOLYL DERIVATIVES EPIX DELAWARE, INC. (US) 2007-04-26 WO disclosed