SCHEMBL5329614

SCHEMBL5329614

COc1cc(F)cc(SC)c1C(N)=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 2/20 0.47
AR P10275 2/20 0.45
SLC6A9 P48067 2/20 0.39
POLB P06746 3/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
KDM4E B2RXH2 1/20 0.37
CTDSP1 Q9GZU7 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
MKNK2 Q9HBH9 1/20 0.35
CSF1R P07333 1/20 0.34
TSHR P16473 2/20 0.34
HTT P42858 2/20 0.34
APOBEC3A P31941 1/20 0.34
APOBEC3G Q9HC16 1/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1349845 0.85 CA12 (0.42) MAP2K1ARSLC6A9POLBKDM4E
SCHEMBL5329932 0.84 SLC6A9 (0.39) MAP2K1ARSLC6A9POLBMEN1
SCHEMBL12439663 0.80 SLC6A9 (0.46) SLC6A9
SCHEMBL5329670 0.78 MAP2K1 (0.50) MAP2K1SLC6A9POLBL3MBTL1KDM4E
SCHEMBL5329470 0.73 CA12 (0.52) ARPOLBL3MBTL1KDM4ECTDSP1
SCHEMBL23327273 0.71 CYP3A4 (0.53) MAP2K1KMT2AALDH1A1RAB9AHTT
SCHEMBL21671633 0.68 CA12 (0.44) MAP2K1L3MBTL1KDM4EALDH1A1RAB9A
SCHEMBL4153927 0.67 CYP3A4 (0.58) POLBL3MBTL1KDM4ECTDSP1TDP1
SCHEMBL11850840 0.67 TSHR (0.59) POLBL3MBTL1KDM4ECTDSP1TDP1
SCHEMBL1004368 0.67 ACHE (0.48) POLBL3MBTL1KDM4ECTDSP1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007147834-A1 GLYCINE TRANSPORTER INHIBITING COMPOUNDS AND USES IN MEDICINE GLAXO GROUP LIMITED (GB) 2007-12-27 WO disclosed