SCHEMBL532963

SCHEMBL532963

Cc1cc(C)c(N2CCCC2)c(C)c1NC(=O)c1ccccc1OCc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SGMS2 Q8NHU3 5/20 0.52
MEN1 O00255 5/20 0.50
KMT2A Q03164 5/20 0.50
GAA P10253 1/20 0.49
LRRK2 Q5S007 2/20 0.48
ALDH1A1 P00352 1/20 0.47
MET P08581 3/20 0.46
POLB P06746 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
NPC1 O15118 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL534153 0.85 MAPT (0.58) MEN1KMT2AALDH1A1POLBSMN1; SMN2
SCHEMBL533022 0.84 MEN1 (0.52) MEN1KMT2AGAASMN1; SMN2NPC1
SCHEMBL534076 0.82 POLB (0.53) MEN1KMT2AGAAALDH1A1POLB
SCHEMBL533064 0.81 MAPT (0.56) MEN1KMT2AGAAALDH1A1POLB
SCHEMBL532973 0.80 MAPT (0.44) MEN1KMT2AGAAALDH1A1POLB
SCHEMBL532826 0.79 ALDH1A1 (0.47) GAAALDH1A1POLBSMN1; SMN2NPSR1
SCHEMBL532801 0.79 GAA (0.48) MEN1KMT2AGAAALDH1A1SMN1; SMN2
SCHEMBL532964 0.79 L3MBTL1 (0.47) MEN1KMT2AGAAALDH1A1SMN1; SMN2
SCHEMBL532950 0.79 KMT2A (0.56) MEN1KMT2AGAAALDH1A1SMN1; SMN2
SCHEMBL533514 0.78 RAB9A (0.51) MEN1KMT2AGAAALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2415760-A2 CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2012-02-08 EP disclosed
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed