SCHEMBL5330447

SCHEMBL5330447

COc1ccccc1C1(O)CCN(CCCN2C(=O)C3CC=CCC3C2=O)CC1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A1 P30531 1/20 0.60
SLC6A12 P48065 1/20 0.60
SLC6A11 P48066 1/20 0.60
SLC6A13 Q9NSD5 1/20 0.60
HSD17B10 Q99714 2/20 0.49
USP2 O75604 1/20 0.49
OPRM1 P35372 1/20 0.45
OPRD1 P41143 1/20 0.45
OPRK1 P41145 1/20 0.45
OPRL1 P41146 1/20 0.45
DRD2 P14416 3/20 0.44
DRD3 P35462 2/20 0.44
ADRA1D P25100 2/20 0.43
ADRA1A P35348 2/20 0.43
ADRA1B P35368 2/20 0.43
SIGMAR1 Q99720 1/20 0.43
POLB P06746 1/20 0.42
HTR1A P08908 3/20 0.42
HTR7 P34969 2/20 0.42
MEN1 O00255 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5592141 0.84 SLC6A1 (0.65) SLC6A1SLC6A12SLC6A11SLC6A13OPRM1
Hydrochloric Acid SCHEMBL5592234 0.83 SLC6A1 (0.64) SLC6A1SLC6A12SLC6A11SLC6A13OPRM1
SCHEMBL5329926 0.82 USP2 (0.48) SLC6A1SLC6A12SLC6A11SLC6A13HSD17B10
SCHEMBL5592122 0.82 SLC6A1 (0.63) SLC6A1SLC6A12SLC6A11SLC6A13OPRM1
Hydrochloric Acid SCHEMBL5592131 0.81 SLC6A1 (0.62) SLC6A1SLC6A12SLC6A11SLC6A13OPRM1
SCHEMBL6240084 0.78 DRD2 (0.71) HSD17B10DRD2DRD3ADRA1DADRA1A
SCHEMBL11808412 0.78 DRD2 (0.66) SLC6A1SLC6A12SLC6A11SLC6A13HSD17B10
Hydrochloric Acid SCHEMBL7105041 0.78 DRD2 (0.70) HSD17B10DRD2DRD3ADRA1DADRA1A
Hydrochloric Acid SCHEMBL11254208 0.76 HTR1A (0.67) SLC6A1SLC6A12SLC6A11SLC6A13DRD2
SCHEMBL6474802 0.75 DRD2 (0.49) HSD17B10USP2DRD2DRD3ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007029156-A2 ISOINDOLEDIONE DERIVATIVES AS ADRENERGIC RECEPTOR ANTAGONISTS RANBAXY LABORATORIES LIMITED (IN) 2007-03-15 WO claimed
WO-2007029156-A2 ISOINDOLEDIONE DERIVATIVES AS ADRENERGIC RECEPTOR ANTAGONISTS RANBAXY LABORATORIES LIMITED (IN) 2007-03-15 WO disclosed