SCHEMBL5330480

SCHEMBL5330480

C=CCCn1c(=O)cc(-c2ccc(C)cc2)n(-c2ccc(SC)cc2)c1=O

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.36
HTT P42858 2/20 0.34
CYP2C9 P11712 1/20 0.34
PTGS2 P35354 8/20 0.34
PTGS1 P23219 2/20 0.32
ADORA2A P29274 1/20 0.31
ADORA2B P29275 1/20 0.31
GSK3A P49840 1/20 0.31
GSK3B P49841 1/20 0.31
CHRNA7 P36544 1/20 0.31
LMNA P02545 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14624154 0.89 THRB (0.37) THRBHTTCYP2C9PTGS2PTGS1
SCHEMBL5325697 0.84 RAD51 (0.40) THRBHTTCYP2C9PTGS2PTGS1
SCHEMBL5320985 0.83 PTGS2 (0.43) THRBHTTCYP2C9PTGS2PTGS1
SCHEMBL5331474 0.83 PTGS2 (0.38) THRBHTTCYP2C9PTGS2PTGS1
SCHEMBL5328124 0.82 PTGS2 (0.37) THRBHTTCYP2C9PTGS2PTGS1
SCHEMBL5324453 0.82 CSF1R (0.40) THRBHTTCYP2C9PTGS2PTGS1
SCHEMBL5320843 0.81 DRD2 (0.44) THRBHTTPTGS2PTGS1LMNA
SCHEMBL5325596 0.80 MEN1 (0.41) HTT
SCHEMBL5296183 0.80 POLB (0.34) THRBHTTCYP2C9PTGS2PTGS1
SCHEMBL14624160 0.80 HTT (0.35) THRBHTTCYP2C9PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007007161-A2 NOVEL BIO-ACTIVE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-01-18 WO claimed
WO-2007007161-A2 NOVEL BIO-ACTIVE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-01-18 WO disclosed
WO-2007007161-A2 NOVEL BIO-ACTIVE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-01-18 WO disclosed