SCHEMBL5296183

SCHEMBL5296183

CSc1ccc(-n2c(-c3ccc(C)cc3)cc(=O)n(CCCCC#N)c2=O)cc1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.34
PTGS2 P35354 7/20 0.33
PTGS1 P23219 2/20 0.33
THRB P10828 1/20 0.32
CYP2C9 P11712 1/20 0.32
HTT P42858 1/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
TDP1 Q9NUW8 1/20 0.32
GRIA2 P42262 1/20 0.32
KMT2A Q03164 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MEN1 O00255 1/20 0.31
GAA P10253 1/20 0.31
HPGD P15428 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5320985 0.85 PTGS2 (0.43) PTGS2PTGS1THRBCYP2C9HTT
SCHEMBL5324453 0.83 CSF1R (0.40) PTGS2PTGS1THRBCYP2C9HTT
SCHEMBL5332569 0.83 MMP2 (0.39) CYP2C9HTTALDH1A1TDP1KMT2A
SCHEMBL5325697 0.81 RAD51 (0.40) PTGS2PTGS1THRBCYP2C9HTT
SCHEMBL5331474 0.80 PTGS2 (0.38) PTGS2PTGS1THRBCYP2C9HTT
SCHEMBL5330480 0.80 THRB (0.36) PTGS2PTGS1THRBCYP2C9HTT
SCHEMBL14624160 0.80 HTT (0.35) POLBPTGS2PTGS1THRBCYP2C9
SCHEMBL5328124 0.79 PTGS2 (0.37) POLBPTGS2PTGS1THRBCYP2C9
SCHEMBL14622453 0.79 CYP11B1 (0.43) POLBHTTKDM4EALDH1A1GAA
SCHEMBL5320843 0.78 DRD2 (0.44) PTGS2PTGS1THRBHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007007161-A2 NOVEL BIO-ACTIVE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-01-18 WO claimed
WO-2007007161-A2 NOVEL BIO-ACTIVE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-01-18 WO disclosed