SCHEMBL5331437

SCHEMBL5331437

CNC(=O)c1ccc(C[As](C)C(=O)C23CC4CC(CC(C4)C2)C3)s1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.37
GPR55 Q9Y2T6 1/20 0.37
NPC1 O15118 3/20 0.36
HPGD P15428 3/20 0.36
RAB9A P51151 3/20 0.36
TP53 P04637 1/20 0.36
TSHR P16473 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HSD11B1 P28845 5/20 0.35
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.35
SMYD3 Q9H7B4 1/20 0.34
CYP3A4 P08684 1/20 0.34
HDAC8 Q9BY41 2/20 0.34
KMT2A Q03164 3/20 0.33
POLB P06746 2/20 0.33
HSD17B10 Q99714 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3323602 0.76 HSD11B1 (0.58) PARP1GPR55HSD11B1CYP3A4KMT2A
SCHEMBL4084359 0.76 ALDH1A1 (0.46) PARP1GPR55NPC1HPGDRAB9A
SCHEMBL12319896 0.68 HSD11B1 (0.59) HPGDTSHRHSD11B1ALDH1A1HDAC8
SCHEMBL11471858 0.67 HPGD (0.50) PARP1NPC1HPGDRAB9ATP53
SCHEMBL12181191 0.67 RAB9A (0.58) PARP1NPC1HPGDRAB9ATP53
SCHEMBL12216734 0.64 KDM4E (0.62) NPC1HPGDRAB9ATSHRSMN1; SMN2
SCHEMBL3749708 0.63 P2RX7 (0.51) ALDH1A1KMT2AHSD17B10MEN1
SCHEMBL24667217 0.63 HPGD (0.46) PARP1NPC1HPGDRAB9ATP53
SCHEMBL28311788 0.62 HPGD (0.57) PARP1NPC1HPGDRAB9ATP53
SCHEMBL29599185 0.62 ALDH1A1 (0.53) PARP1NPC1HPGDRAB9ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1861384-A1 11-BETA-HYDROXYSTEROID DEHYDROGENASE INHIBITORS Sterix Limited (GB) 2007-12-05 EP disclosed
WO-2006100502-A1 11-BETA-HYDROXYSTEROID DEHYDROGENASE INHIBITORS STERIX LIMITED (GB) 2006-09-28 WO disclosed