SCHEMBL5331579

SCHEMBL5331579

COc1ccc(CNC(=O)/C=C\C(=O)N2CCN(C(c3ccccc3)c3ccc(Cl)cc3)CC2)cc1

nearest known ligand 0.64

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CACNA1G O43497 6/20 0.64
GPX4 P36969 1/20 0.59
LMNA P02545 1/20 0.59
TACR3 P29371 1/20 0.56
CACNA2D1 P54289 8/20 0.53
CACNB1 Q02641 8/20 0.53
CACNA1B Q00975 6/20 0.53
CACNA1C Q13936 5/20 0.53
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
MAPT P10636 1/20 0.50
CACNA1A O00555 2/20 0.48
TDP1 Q9NUW8 1/20 0.47
DRD2 P14416 1/20 0.47
DRD3 P35462 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5351830 0.90 TACR3 (0.59) CACNA1GGPX4TACR3CACNA2D1CACNB1
SCHEMBL5326872 0.90 TACR3 (0.59) CACNA1GGPX4TACR3CACNA2D1CACNB1
SCHEMBL5365428 0.87 LMNA (0.52) CACNA1GGPX4LMNACACNA2D1CACNB1
SCHEMBL5357281 0.87 LMNA (0.52) CACNA1GGPX4LMNACACNA2D1CACNB1
SCHEMBL5329966 0.80 CACNA1G (0.67) CACNA1GLMNACACNA2D1CACNB1CACNA1B
SCHEMBL5372531 0.80 CACNA1G (0.66) CACNA1GLMNACACNA2D1CACNB1CACNA1B
SCHEMBL5324722 0.78 TACR3 (0.58) CACNA1GGPX4LMNATACR3CACNA2D1
SCHEMBL5362020 0.78 CACNA1G (0.63) CACNA1GLMNACACNA2D1CACNB1CACNA1B
SCHEMBL5329875 0.76 CA1 (0.50) GPX4LMNACACNA2D1CACNB1CACNA1B
SCHEMBL16598473 0.75 TACR3 (0.67) CACNA1GTACR3CACNA2D1CACNB1CACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007142431-A1 NEW NON-PEPTIDE COMPOUNDS, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME EWHA UNIVERSITY - INDUSTRY COLLABORATION FOUNDATION (KR) 2007-12-13 WO disclosed
WO-2007142431-A1 NEW NON-PEPTIDE COMPOUNDS, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME EWHA UNIVERSITY - INDUSTRY COLLABORATION FOUNDATION (KR) 2007-12-13 WO disclosed