Tetrazole

Tetrazole

SCHEMBL5331869

Cc1ccccc1-c1ccccc1.c1nnn[nH]1

nearest known ligand 0.42

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP3 O14638 1/20 0.42
ENPP1 P22413 1/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
GAA P10253 1/20 0.39
DCUN1D1 Q96GG9 2/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
KDM4E B2RXH2 1/20 0.37
AKT1 P31749 1/20 0.37
AKT2 P31751 1/20 0.37
ESR2 Q92731 1/20 0.37
TRPA1 O75762 1/20 0.36
CASP3 P42574 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Biphenyl SCHEMBL9308 0.81 ALDH1A1 (0.43) NPC1RAB9ASMN1; SMN2ALDH1A1HPGD
Biphenyl SCHEMBL28349299 0.80 AKT2 (0.38) ALDH1A1KDM4EAKT1AKT2IDO1
Biphenyl SCHEMBL28359469 0.80 ALDH1A1 (0.38) NPC1RAB9ASMN1; SMN2ALDH1A1KDM4E
Tetrazole SCHEMBL28778836 0.79 ALDH1A1 (0.59) NPC1RAB9ASMN1; SMN2ALDH1A1HPGD
Tetrazole SCHEMBL27729626 0.79 ALDH1A1 (0.59) NPC1RAB9ASMN1; SMN2ALDH1A1HPGD
Biphenyl SCHEMBL1627148 0.79 ALDH1A1 (0.41) NPC1RAB9ASMN1; SMN2ALDH1A1HPGD
Tetrazole SCHEMBL29023855 0.79 ALDH1A1 (0.41) NPC1RAB9ASMN1; SMN2ALDH1A1HPGD
Biphenyl SCHEMBL27802159 0.79 ALDH1A1 (0.41) NPC1RAB9ASMN1; SMN2ALDH1A1HPGD
Biphenyl SCHEMBL9158420 0.79 ALDH1A1 (0.41) NPC1RAB9ASMN1; SMN2ALDH1A1HPGD
Tetrazole SCHEMBL28320883 0.79 NPC1 (0.43) NPC1RAB9ASMN1; SMN2ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0971747-B1 CONTRAST AGENTS AMERSHAM HEALTH AS (NO) 2005-12-28 EP claimed
US-6921525-B2 Contrast agents AMERSHAM HEALTH AS (NO) 2005-07-26 US claimed
US-20030228254-A1 Diagnosis of cardiovascular disorders AMERSHAM HEALTH AS (NO) 2003-12-11 US claimed
US-20010016587-A1 Contrast agents NYCOMED IMAGING AS 2001-08-23 US claimed
EP-0971747-A2 CONTRAST AGENTS NYCOMED IMAGING AS (NO) 2000-01-19 EP claimed
CN-101480390-A Compound preparation containing Sartan and diuretics BEIJING INST TECHNOLOGY (CN) 2009-07-15 CN disclosed
CN-101361736-A Compound of losartan or pharmaceutical salt thereof and calcium channel blockers or pharmaceutical salt thereof BEIJING INST TECHNOLOGY (CN) 2009-02-11 CN disclosed
CN-101347427-A Compound of losartan compound or its medical salt and calcium channel blocker or its medical salt BEIJING INST TECHNOLOGY (CN) 2009-01-21 CN disclosed
US-7182934-B2 Ultrasonic contrast agents; aqueous suspension GE HEALTHCARE AS (NO) 2007-02-27 US disclosed
EP-0971747-B1 CONTRAST AGENTS AMERSHAM HEALTH AS (NO) 2005-12-28 EP disclosed
US-20050201930-A1 Contrast agents GE HEALTHCARE AS (NO) 2005-09-15 US disclosed
US-6921525-B2 Contrast agents AMERSHAM HEALTH AS (NO) 2005-07-26 US disclosed
US-20030228254-A1 Diagnosis of cardiovascular disorders AMERSHAM HEALTH AS (NO) 2003-12-11 US disclosed
US-6524552-B2 Imaging cardiovascular disorders GE HEALTHCARE AS (NO) 2003-02-25 US disclosed
US-20010016587-A1 Contrast agents NYCOMED IMAGING AS 2001-08-23 US disclosed
US-6264914-B1 CONTAINING IMIDAZOLE RING NYCOMED IMAGING AS (NO) 2001-07-24 US disclosed
EP-0971747-A2 CONTRAST AGENTS NYCOMED IMAGING AS (NO) 2000-01-19 EP disclosed
WO-1998018496-A2 CONTRAST AGENTS NYCOMED IMAGING AS (NO) 1998-05-07 WO disclosed
CN-1123276-A Cycloheptimidazole derivatives, method of manufacturing the same and therapeutic agents containing these compounds KOTOBUKI SEIYAKU CO LTD (JP) 1996-05-29 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030228254-A1 Diagnosis of cardiovascular disorders AGTR1, AGTR2, AGT ENPP3 3419/4885ENPP1 3540/4885NPC1 2884/4885
US-20010016587-A1 Contrast agents AGTR1, AGTR2, VIPR1 ENPP3 3400/4885ENPP1 3492/4885NPC1 1915/4885
US-20050201930-A1 Contrast agents AGTR1, AGTR2, VIPR1 ENPP3 2649/4885ENPP1 3124/4885NPC1 2481/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.