SCHEMBL5332136

SCHEMBL5332136

CC(C)(C)[Si](C)(C)OCc1cc(-c2ccc(F)cc2C(F)(F)F)no1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.38
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
KCNH2 Q12809 1/20 0.37
GRM5 P41594 6/20 0.34
AR P10275 4/20 0.33
POLB P06746 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
TRPA1 O75762 1/20 0.32
CACNA1G O43497 1/20 0.32
P2RX7 Q99572 1/20 0.31
WDR5 P61964 1/20 0.31
CASP3 P42574 1/20 0.31
SENP8 Q96LD8 1/20 0.31
SENP7 Q9BQF6 1/20 0.31
SENP6 Q9GZR1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5331359 0.84 NPC1 (0.38) NPC1RAB9AKCNH2POLBSMN1; SMN2
SCHEMBL542216 0.79 KCNH2 (0.42) IDO1NPC1RAB9AKCNH2GRM5
SCHEMBL5309293 0.78 NOTUM (0.45) IDO1NPC1RAB9AKCNH2AR
SCHEMBL5327885 0.74 RAB9A (0.45) NPC1RAB9APOLBSMN1; SMN2L3MBTL1
SCHEMBL15084169 0.74 NTRK1 (0.40) NPC1RAB9AARTRPA1P2RX7
SCHEMBL5802338 0.71 L3MBTL1 (0.38) NPC1RAB9APOLBSMN1; SMN2L3MBTL1
SCHEMBL5802677 0.71 AR (0.33) KCNH2ARTRPA1
SCHEMBL3721862 0.69 CACNA1G (0.42) NPC1RAB9AKCNH2SMN1; SMN2CACNA1G
SCHEMBL1220435 0.69 MAPT (0.41) NPC1RAB9APOLBSMN1; SMN2L3MBTL1
SCHEMBL5332143 0.69 GALR3 (0.34) IDO1GRM5ARSMN1; SMN2TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007034445-A2 NOVEL PIPERAZINE DERIVATIVES AS RENIN INHIBITORS FOR CARDIOVASCULAR EVENTS AND RENAL INSUFFICIENCY ACTELION PHARMACEUTICALS LTD (CH) 2007-03-29 WO disclosed
WO-2006064484-A1 AZABICYCLONONENE DERIVATIVES AS RENIN INHIBITORS ACTELION PHARMACEUTICALS LTD (CH) 2006-06-22 WO disclosed