SCHEMBL5331359

SCHEMBL5331359

CC(C)(C)[Si](C)(C)OCc1cc(-c2ccc(F)cc2Cl)no1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.38
RAB9A P51151 6/20 0.38
CNR1 P21554 3/20 0.38
CNR2 P34972 3/20 0.38
MAPT P10636 6/20 0.36
ALDH1A1 P00352 2/20 0.36
PKM P14618 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
CYP3A4 P08684 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTT P42858 1/20 0.35
RECQL P46063 1/20 0.35
L3MBTL1 Q9Y468 3/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
POLB P06746 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
REN P00797 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5327885 0.88 RAB9A (0.45) NPC1RAB9AMAPTALDH1A1PKM
SCHEMBL5332136 0.84 IDO1 (0.38) NPC1RAB9AL3MBTL1SMN1; SMN2POLB
SCHEMBL5334510 0.77 CHRNB2 (0.38) NPC1RAB9AMAPTALDH1A1CHRNB2
SCHEMBL5335644 0.77 MAPT (0.40) NPC1RAB9AMAPTALDH1A1CYP3A4
SCHEMBL5802338 0.77 L3MBTL1 (0.38) NPC1RAB9AMAPTL3MBTL1SMN1; SMN2
SCHEMBL5306222 0.76 NOTUM (0.53) NPC1RAB9AMAPTALDH1A1PKM
SCHEMBL5802048 0.70 CNR2 (0.35) NPC1RAB9ACNR1CNR2MAPT
SCHEMBL23982537 0.68 CHRNB2 (0.46) NPC1RAB9AMAPTALDH1A1PKM
SCHEMBL5331361 0.68 CNR2 (0.38) NPC1RAB9ACNR1CNR2MAPT
SCHEMBL3759539 0.67 MEN1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007034445-A2 NOVEL PIPERAZINE DERIVATIVES AS RENIN INHIBITORS FOR CARDIOVASCULAR EVENTS AND RENAL INSUFFICIENCY ACTELION PHARMACEUTICALS LTD (CH) 2007-03-29 WO disclosed
WO-2006064484-A1 AZABICYCLONONENE DERIVATIVES AS RENIN INHIBITORS ACTELION PHARMACEUTICALS LTD (CH) 2006-06-22 WO disclosed