SCHEMBL5333323

SCHEMBL5333323

C=CCc1c(N)ccc(-c2ccc(N)c(CC=C)c2CC=C)c1CC=C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 1/20 0.49
ALDH1A1 P00352 3/20 0.33
GABRA1 P14867 2/20 0.33
GABRB2 P47870 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH2 P05091 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
AKR1B1 P15121 1/20 0.33
HPGD P15428 1/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
PPARG P37231 1/20 0.33
KMT2A Q03164 1/20 0.33
PPARD Q03181 1/20 0.33
XDH P47989 1/20 0.30
TP53 P04637 1/20 0.30
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10885430 0.98 IMPDH2 (0.47) IMPDH2ALDH1A1GABRA1GABRB2NPSR1
SCHEMBL845635 0.93 IMPDH2 (0.53) IMPDH2ALDH1A1GABRA1GABRB2NPSR1
SCHEMBL1334154 0.84 IMPDH2 (0.41) IMPDH2ALDH1A1GABRA1GABRB2KDM4E
SCHEMBL2358033 0.82 IMPDH2 (0.46) IMPDH2GABRA1GABRB2NPSR1
SCHEMBL6139914 0.80 IMPDH2 (0.45) IMPDH2GABRA1GABRB2
Water SCHEMBL11758577 0.80 IMPDH2 (0.45) IMPDH2GABRA1GABRB2
SCHEMBL4976094 0.80 IMPDH2 (0.45) IMPDH2ALDH1A1NPSR1MAPTTP53
SCHEMBL6572591 0.80 SRD5A1 (0.45) IMPDH2ALDH1A1GABRA1GABRB2NPSR1
SCHEMBL10709835 0.78 IMPDH2 (0.46) IMPDH2ALDH1A1GABRA1GABRB2NPSR1
SCHEMBL10879094 0.77 IMPDH2 (0.42) IMPDH2NPSR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 75 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0918881-B1 DRY REAGENT TEST STRIP COMPRISING BENZIDINE DYE PRECURSOR AND ANTIPYRINE COMPOUND AMIRA MEDICAL (US) 2004-02-11 EP claimed
WO-2000039586-A2 TETRAMETHYLBENZIDINE FORMULATION FOR HORSERADISH PEROXIDASE ENZYME ASSAYS SEDUM LABORATORIES (US) 2000-07-06 WO claimed
EP-0918881-A1 DRY REAGENT TEST STRIP COMPRISING BENZIDINE DYE PRECURSOR AND ANTIPYRINE COMPOUND Mercury Diagnostics Inc. (US) 1999-06-02 EP claimed
US-5824491-A OXIDASE ENZYME AS ANALYTE ON SUBSTRATE, FORMING PEROXIDE, BENZIDINE DYE PRECURSOR, PEROXIDASE ENZYME WITH ANTIPYRENE COMPOUND MERCURY DIAGNOSTICS, INC. (US) 1998-10-20 US claimed
WO-1997044482-A1 DRY REAGENT TEST STRIP COMPRISING BENZIDINE DYE PRECURSOR AND ANTIPYRINE COMPOUND MERCURY DIAGNOSTICS INC. (US) 1997-11-27 WO claimed
US-5610026-A OF AN AQUEOUS SOLUTION CONTAINING A TETRAALKYLBENZIDINE OR A SALT THEREOF, A PEROXIDE OR A SYSTEM GENERATING HYDROGEN PEROXIDE AND A BUFFER BEHRINGWERKE AKTIENGESELLSCHAFT (DE) 1997-03-11 US claimed
US-5491094-A COLORIMETRIC ANALYSIS INDICATOR 3,3*,5,5*-TETRAALKYLBENZIDINE INDUSTRIAL TEST SYSTEMS, INC. (US) 1996-02-13 US claimed
US-5206150-A Tetramethylbenzidine, peroxide and bacitracin as stabilizer; incubation UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 1993-04-27 US claimed
EP-0224813-B1 MEANS FOR DETECTING PEROXIDASE ACTIVITY WITH A STABILIZER, PREPARATION PROCESS AND ITS USE BEHRINGWERKE Aktiengesellschaft (DE) 1990-09-26 EP claimed
EP-0224210-B1 MEANS FOR DETECTING PEROXIDASE ACTIVITY, PREPARATION PROCESS AND ITS USE BEHRINGWERKE Aktiengesellschaft (DE) 1990-08-29 EP claimed
US-4891314-A STORAGE STABILITY BEHRINGWERKE AKTIENGESELLSCHAFT (DE) 1990-01-02 US claimed
US-4562148-A IMMUNOASSAY, CARBOXYLATE OR SULFONATE POLYMER MILES LABORATORIES, INC. (US) 1985-12-31 US claimed
JP-1104196-A None JP disclosed
JP-8080199-A None JP disclosed
JP-61052300-A None JP disclosed
JP-8313525-A None JP disclosed
US-4385114-A DETERMINATION OF HYDROGEN PEROXIDE OR PEROXIDASE BOEHRINGER MANNHEIM GMBH (DE) 1983-05-24 US disclosed
EP-0078965-A1 Method for preparing an analytical element preventing reagent migration MILES LABORATORIES, INC. (US) 1983-05-18 EP disclosed
EP-0071934-A1 Method for preparing a color stable chromogenic analytical element MILES LABORATORIES, INC. (US) 1983-02-16 EP disclosed
US-4361648-A POLYMERIC MORDANT, TETRAALKYLBENZIDINE HYDROCHLORIDE, ENZYME, PEROXIDATIVELY ACTIVE MATERIAL MILES LABORATORIES, INC. (US) 1982-11-30 US disclosed