SCHEMBL5333969

SCHEMBL5333969

Cn1cc([N+](=O)[O-])cc1-c1nc2cc(C(=O)O)ccc2[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 5/20 0.47
KMT2A Q03164 5/20 0.47
MEN1 O00255 4/20 0.47
MAPT P10636 4/20 0.47
POLB P06746 1/20 0.47
NPC1 O15118 4/20 0.47
RAB9A P51151 4/20 0.47
NPBWR1 P48145 2/20 0.44
HSP90AA1 P07900 1/20 0.40
ESR2 Q92731 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
MMP2 P08253 2/20 0.38
MMP9 P14780 2/20 0.38
MMP8 P22894 2/20 0.38
MMP13 P45452 2/20 0.38
CHRM4 P08173 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8601049 0.91 CHEK2 (0.58) CHEK2KMT2AMEN1MAPTPOLB
SCHEMBL5559865 0.88 MEN1 (0.47) CHEK2KMT2AMEN1MAPTPOLB
SCHEMBL14224669 0.85 MEN1 (0.49) KMT2AMEN1MAPTPOLBNPC1
SCHEMBL8601035 0.83 KMT2A (0.43) CHEK2KMT2AMEN1MAPTPOLB
SCHEMBL7471355 0.83 MAPT (0.43) KMT2AMEN1MAPTPOLBNPC1
SCHEMBL7473157 0.81 MAPT (0.43) KMT2AMEN1MAPTPOLBNPC1
SCHEMBL7465939 0.80 MAPT (0.43) KMT2AMEN1MAPTPOLBNPC1
SCHEMBL7470258 0.80 HPGD (0.46) KMT2AMEN1MAPTPOLBNPC1
SCHEMBL7470356 0.80 TDP1 (0.48) CHEK2KMT2AMEN1MAPTPOLB
SCHEMBL15233046 0.80 IRAK4 (0.54) CHEK2KMT2AMEN1MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007045096-A1 OLIGOHETEROAROMATIC LUMINISCENT ASSEMBLIES AS HIGH-AFFINITY DNA SEQUENCE-DIRECTED LIGANDS UNIVERSITY OF SASKATCHEWAN (CA) 2007-04-26 WO disclosed
EP-0711768-B1 BENZIMIDAZOLE DERIVATIVE MITSUI CHEMICALS INC (JP) 2002-02-13 EP disclosed
EP-0776891-B1 Pyrrolylbenzimidazole derivatives MITSUI CHEMICALS INC (JP) 1999-02-10 EP disclosed
US-5852011-A Benzimidazole derivatives MITSUI CHEMICALS, INC. (JP) 1998-12-22 US disclosed
US-5808087-A ANTITUMOR, ANTICANCER AGENTS MITSUI CHEMICALS, INC. (JP) 1998-09-15 US disclosed
EP-0776891-A1 Pyrrolylbenzimidazole derivatives MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1997-06-04 EP disclosed
EP-0711768-A1 BENZIMIDAZOLE DERIVATIVE MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-05-15 EP disclosed