SCHEMBL5336795

SCHEMBL5336795

CNc1nc(-c2ccccc2)ccc1C#N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.52
ALDH1A1 P00352 7/20 0.52
HPGD P15428 3/20 0.52
GAA P10253 3/20 0.52
MAPT P10636 5/20 0.50
CYP1A2 P05177 3/20 0.50
CYP3A4 P08684 3/20 0.50
CYP2C19 P33261 3/20 0.50
CYP2C9 P11712 2/20 0.50
KMT2A Q03164 8/20 0.48
MEN1 O00255 7/20 0.48
L3MBTL1 Q9Y468 2/20 0.47
ADORA1 P30542 2/20 0.45
ADORA2A P29274 1/20 0.45
NPSR1 Q6W5P4 1/20 0.43
TDP1 Q9NUW8 3/20 0.43
LMNA P02545 1/20 0.43
GLA P06280 1/20 0.42
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5338895 0.84 NLRP3 (0.51) KDM4EALDH1A1HPGDGAAMAPT
SCHEMBL27241714 0.79 MAPT (0.51) KDM4EALDH1A1HPGDGAAMAPT
SCHEMBL17819123 0.77 ALOX15 (0.51) KDM4EALDH1A1HPGDGAAMAPT
SCHEMBL24154751 0.76 KMT2A (0.56) KDM4EALDH1A1HPGDGAAMAPT
SCHEMBL30319960 0.76 KMT2A (0.56) KDM4EALDH1A1HPGDGAAMAPT
SCHEMBL7219112 0.75 ADORA1 (0.53) KDM4EALDH1A1HPGDMAPTCYP1A2
SCHEMBL5329336 0.74 ADORA1 (0.56) KDM4EALDH1A1HPGDGAAMAPT
SCHEMBL1904903 0.74 CYP1A2 (0.53) KDM4EALDH1A1HPGDMAPTCYP1A2
SCHEMBL7834299 0.74 MAP2K3 (0.49) KDM4EALDH1A1HPGDGAAMAPT
SCHEMBL19805092 0.74 MEN1 (0.50) KDM4EALDH1A1HPGDMAPTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007029062-A2 NOVEL PYRIDINE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-03-15 WO claimed