SCHEMBL5339709

SCHEMBL5339709

CCOC(=O)C1=C(C)NC(=O)NC1c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.80

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.68
CA1 P00915 1/20 0.68
CA2 P00918 1/20 0.68
CA7 P43166 1/20 0.68
CA9 Q16790 1/20 0.68
HSD17B10 Q99714 1/20 0.67
MEN1 O00255 1/20 0.65
KMT2A Q03164 1/20 0.65
ADORA3 P0DMS8 1/20 0.63
L3MBTL1 Q9Y468 1/20 0.62
ADORA2B P29275 3/20 0.61
CYP1A2 P05177 1/20 0.61
CYP2C9 P11712 1/20 0.61
MAPK1 P28482 1/20 0.61
CYP2C19 P33261 1/20 0.61
ALDH1A1 P00352 1/20 0.60
EPHX2 P34913 1/20 0.60
KIF11 P52732 1/20 0.60
GAA P10253 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19752618 1.00 CA12 (0.68) CA12CA1CA2CA7CA9
SCHEMBL28346675 0.88 PKM (0.59) KMT2AADORA3L3MBTL1ADORA2BALDH1A1
SCHEMBL3394058 0.86 ALDH1A1 (0.71) MEN1KMT2AADORA3L3MBTL1CYP1A2
SCHEMBL29531249 0.86 ALDH1A1 (0.71) MEN1KMT2AADORA3L3MBTL1CYP1A2
SCHEMBL19752716 0.86 ALDH1A1 (0.71) MEN1KMT2AADORA3L3MBTL1CYP1A2
SCHEMBL1227524 0.85 HSD17B10 (0.77) CA12CA1CA2CA7CA9
SCHEMBL19752680 0.85 HSD17B10 (0.77) CA12CA1CA2CA7CA9
SCHEMBL10112951 0.84 HSD17B10 (0.76) CA12CA1CA2CA7CA9
SCHEMBL5340705 0.84 HSD17B10 (0.75) CA12CA1CA2CA7CA9
SCHEMBL19732962 0.84 ALDH1A1 (0.55) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114740098-B Application of chiral Cd-MOFs material in resolution of dihydropyrimidinone derivative in high performance liquid chromatography 兰州大学 2023-08-01 CN disclosed
CN-112812066-B Synthesis method of dihydropyrimidinone compound 宜春学院 2023-04-25 CN disclosed
CN-114740098-A Application of chiral Cd-MOFs material in resolution of dihydropyrimidinone derivative in high performance liquid chromatography 兰州大学 2022-07-12 CN disclosed
CN-110437100-B Preparation method and application of novel ionic salicylaldehyde Schiff base zirconium complex 山西医科大学 2022-03-11 CN disclosed
CN-112812066-A Synthesis method of dihydropyrimidinone compounds 宜春学院 2021-05-18 CN disclosed
EP-3260446-A1 ENANTIOSELECTIVE SYNTHESIS OF DIHYDROPYRIMIDINONES AND HEXAHYDROPYRIMIDINONES Universitat de les Illes Balears (ES) 2017-12-27 EP disclosed
WO-2007101213-A2 NOVEL 2-OXO-1,2,3,4-TETRAHYDROPYRIMIDINES, BICYCLIC PYRIMIDINE DIONES AND IMIDAZOLIDINE-2,4-DIONES USEFUL AS INDUCIBLE NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2007-09-07 WO disclosed