SCHEMBL534781

SCHEMBL534781

COCc1cc(C(=O)O)ccc1-c1ccccc1C(F)(F)F.COCc1cc(C(=O)O)ccc1-c1ccccc1Cl.COCc1cc(C(=O)O)ccc1-c1ccccc1F.COCc1cc(C(=O)O)ccc1N1CCCC1C.C[C@@H]1CCCCN1c1ccc(C(=O)O)cc1C(F)(F)F.C[C@H]1CCCCN1c1ccc(C(=O)O)cc1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 5/20 0.40
RORC P51449 10/20 0.36
TTR P02766 2/20 0.36
RBP4 P02753 1/20 0.36
NR1H4 Q96RI1 2/20 0.36
PPARG P37231 1/20 0.35
RARA P10276 1/20 0.34
RARB P10826 1/20 0.34
RARG P13631 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL536094 0.86 PRKG1 (0.38) NR1H4
SCHEMBL536095 0.79 BRD4 (0.35)
SCHEMBL536674 0.78 S1PR1 (0.39) S1PR1
SCHEMBL1725696 0.76 S1PR1 (0.48) S1PR1RORCTTR
SCHEMBL408083 0.76 GFER (0.46) S1PR1
SCHEMBL410352 0.75 GFER (0.42)
SCHEMBL1725667 0.75 S1PR1 (0.48) S1PR1TTRRARARARBRARG
SCHEMBL3466223 0.74 S1PR1 (0.37) S1PR1TTRRBP4RARARARB
SCHEMBL409116 0.74 S1PR1 (0.49) S1PR1TTRRARARARBRARG
SCHEMBL536168 0.74 S1PR1 (0.49) S1PR1TTRRARARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414341-A2 OXADIAZOLE DERIVATIVES Merck Serono SA (CH) 2012-02-08 EP disclosed
WO-2010115751-A2 OXADIAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2010-10-14 WO disclosed