SCHEMBL536674

SCHEMBL536674

COCc1cc(C(=O)O)ccc1-c1ccccc1C.COCc1cc(C(=O)O)ccc1N1CCCCC1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 6/20 0.39
S1PR3 Q99500 2/20 0.39
PLAUR Q03405 1/20 0.38
PLA2G7 Q13093 1/20 0.38
POLB P06746 1/20 0.38
TSHR P16473 1/20 0.38
GFER P55789 1/20 0.38
MAPT P10636 2/20 0.38
KDM4E B2RXH2 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
TPH1 P17752 1/20 0.37
NR1I2 O75469 2/20 0.37
SMARCA2 P51531 2/20 0.37
SMARCA4 P51532 2/20 0.37
NR1H3 Q13133 2/20 0.37
PBRM1 Q86U86 2/20 0.37
NR1H2 P55055 1/20 0.37
CACNA1G O43497 2/20 0.36
NR3C2 P08235 1/20 0.36
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL408083 0.88 GFER (0.46) S1PR1PLAURPOLBGFERKDM4E
SCHEMBL536094 0.87 PRKG1 (0.38) PLAURPOLBTSHRKDM4ENR1I2
SCHEMBL410352 0.85 GFER (0.42) POLBGFERKDM4EL3MBTL1TPH1
SCHEMBL536177 0.84 S1PR1 (0.39) S1PR1S1PR3PLA2G7POLBTSHR
SCHEMBL3466223 0.81 S1PR1 (0.37) S1PR1S1PR3POLBMAPTKDM4E
SCHEMBL319590 0.81 S1PR1 (0.52) S1PR1S1PR3POLB
SCHEMBL536095 0.79 BRD4 (0.35) GFERMAPTKDM4ENR1I2SMARCA2
SCHEMBL534781 0.78 S1PR1 (0.40) S1PR1
SCHEMBL2482448 0.78 S1PR1 (0.35) S1PR1KDM4ENR3C2
SCHEMBL1725667 0.77 S1PR1 (0.48) S1PR1PLAURPLA2G7POLBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414342-A1 OXADIAZOLE DERIVATIVES Merck Serono S.A. (CH) 2012-02-08 EP disclosed
WO-2010112461-A1 OXADIAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2010-10-07 WO disclosed