SCHEMBL536095

SCHEMBL536095

COCc1cc(C(=O)OC(=O)c2ccc(N3CCCC3C)c(COC)c2)ccc1-c1ccccc1Cl

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.35
BRPF1 P55201 2/20 0.35
NR1I2 O75469 2/20 0.35
SMARCA2 P51531 2/20 0.35
SMARCA4 P51532 2/20 0.35
PBRM1 Q86U86 2/20 0.35
NR1H2 P55055 1/20 0.35
HPGD P15428 2/20 0.35
ALOX15 P16050 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CHRM3 P20309 1/20 0.34
NPC1 O15118 1/20 0.34
CASP3 P42574 1/20 0.34
RAB9A P51151 1/20 0.34
SENP8 Q96LD8 1/20 0.34
SENP7 Q9BQF6 1/20 0.34
SENP6 Q9GZR1 1/20 0.34
MAPK14 Q16539 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL536094 0.92 PRKG1 (0.38) BRD4BRPF1NR1I2SMARCA2SMARCA4
SCHEMBL534781 0.79 S1PR1 (0.40)
SCHEMBL536674 0.79 S1PR1 (0.39) NR1I2SMARCA2SMARCA4PBRM1NR1H2
SCHEMBL410352 0.78 GFER (0.42) BRD4BRPF1HPGDALOX15HSD17B10
SCHEMBL406399 0.75 MAPK14 (0.44) HSD17B10NPC1RAB9AMAPK14ALDH1A1
SCHEMBL408083 0.75 GFER (0.46) HPGDHSD17B10KDM4EGAAGFER
SCHEMBL536178 0.72 S1PR1 (0.39) NR1I2SMARCA2SMARCA4PBRM1NR1H2
SCHEMBL406660 0.72 NR4A2 (0.46) HPGDNPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL407058 0.69 AR (0.39) NR1I2SMARCA2SMARCA4PBRM1NR1H2
SCHEMBL410064 0.66 PDK2 (0.45) HPGDHSD17B10NPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414342-A1 OXADIAZOLE DERIVATIVES Merck Serono S.A. (CH) 2012-02-08 EP disclosed
WO-2010112461-A1 OXADIAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2010-10-07 WO disclosed