SCHEMBL5354675

SCHEMBL5354675

Cc1[nH]cc(C(=O)OCc2ccccc2)c1-c1ccc(C#N)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 2/20 0.47
ALDH1A1 P00352 4/20 0.43
TDP1 Q9NUW8 3/20 0.42
MAOB P27338 1/20 0.41
MAPK1 P28482 2/20 0.41
TSHR P16473 2/20 0.41
CYP3A4 P08684 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
RAB9A P51151 4/20 0.40
NPC1 O15118 2/20 0.40
POLB P06746 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
MAPT P10636 1/20 0.40
STAT1 P42224 1/20 0.40
ATM Q13315 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
KMT2A Q03164 2/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A3 Q01959 1/20 0.40
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6464844 0.82 HTT (0.53) ARALDH1A1TDP1MAOBMAPK1
SCHEMBL5359751 0.81 LMNA (0.52) ARALDH1A1MAOBMAPK1RAB9A
SCHEMBL5361928 0.80 AR (0.49) ARALDH1A1TDP1MAOBMAPK1
SCHEMBL6466360 0.80 RAB9A (0.57) ARALDH1A1TDP1MAPK1TSHR
SCHEMBL5360596 0.78 AR (0.47) ARALDH1A1TDP1MAOBMAPK1
SCHEMBL2656845 0.78 CLEC4M (0.46) ALDH1A1CYP3A4NPSR1MAPTATM
SCHEMBL4921544 0.78 RAB9A (0.46) ARALDH1A1TDP1MAPK1TSHR
SCHEMBL4914072 0.77 KDM1A (0.38) AR
SCHEMBL14347608 0.77 ALDH1A1 (0.51) ARALDH1A1MAPK1RAB9ANPC1
SCHEMBL28942197 0.77 ALDH1A1 (0.50) ALDH1A1TDP1MAPK1TSHRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed