SCHEMBL5355017

SCHEMBL5355017

O=c1[nH]nc2cnc3ccc(F)cc3n12

nearest known ligand 0.59

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 10/20 0.40
NOTUM Q6P988 2/20 0.38
JAK2 O60674 2/20 0.36
JAK3 P52333 2/20 0.36
GRM2 Q14416 2/20 0.36
DAO P14920 1/20 0.36
PARP1 P09874 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL796231 0.82 CHEK1 (0.58) CHEK1
SCHEMBL5362675 0.82 ADORA3 (0.43) CHEK1NOTUM
SCHEMBL560634 0.78 MAPT (0.54) CHEK1DAO
SCHEMBL5479035 0.72 CHEK1 (0.68) CHEK1
SCHEMBL18544256 0.71 PARP1 (0.38) DAOPARP1
SCHEMBL5732439 0.69 PDE2A (0.38) GRM2
SCHEMBL19231294 0.67 CYP11B1 (0.44) PARP1
SCHEMBL5349697 0.65 HRH4 (0.38)
SCHEMBL5357419 0.65 ADORA1 (0.44)
SCHEMBL8910786 0.65 DAO (0.49) GRM2DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7202245-B2 Substituted 4-amino[1,2,4]triazolo[4,3-a] quinoxalines PFIZER INC. (US) 2007-04-10 US disclosed