SCHEMBL5355040

SCHEMBL5355040

Cc1cc2c(cc1COc1ccccc1)C(C1CCCCC1)=NN(C)C(=O)N2

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTH1R Q03431 5/20 0.39
ADAM17 P78536 2/20 0.36
BRD4 O60885 1/20 0.35
IDH1 O75874 1/20 0.35
ALDH1A1 P00352 2/20 0.34
CCKBR P32239 2/20 0.34
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
CD274 Q9NZQ7 1/20 0.34
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
CCKAR P32238 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5362739 0.81 PTH1R (0.35) PTH1RCCKBRCCKAR
SCHEMBL5326023 0.77 PTH1R (0.37) PTH1RBRD4CCKBR
SCHEMBL5355357 0.77 BRD4 (0.36) PTH1RBRD4ALDH1A1CCKBR
SCHEMBL5355360 0.77 BRD4 (0.36) PTH1RBRD4ALDH1A1CCKBR
SCHEMBL5358455 0.76 BCHE (0.37) PTH1RALDH1A1CCKBR
SCHEMBL5321928 0.76 ALDH1A1 (0.35) PTH1RALDH1A1CCKBR
SCHEMBL5355386 0.74 ALDH1A1 (0.36) PTH1RALDH1A1PDE4APDE4BPDE4C
SCHEMBL5329713 0.73 PTH1R (0.45) PTH1RALDH1A1CCKBR
SCHEMBL5353466 0.72 PTH1R (0.54) PTH1R
SCHEMBL5323349 0.72 ALDH1A1 (0.34) PTH1RALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007135417-A1 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2007-11-29 WO disclosed