SCHEMBL5358282

SCHEMBL5358282

Cc1[nH]c(C#N)c(C)c1-c1ccc(C#N)c(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 5/20 0.41
TRPV4 Q9HBA0 1/20 0.40
NSD2 O96028 1/20 0.40
AR P10275 5/20 0.38
CYP11B1 P15538 3/20 0.37
GRIA1 P42261 1/20 0.37
CACNG8 Q8WXS5 1/20 0.37
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
CASP1 P29466 1/20 0.36
EGLN2 Q96KS0 1/20 0.36
DAO P14920 1/20 0.34
CDK4 P11802 1/20 0.34
CDK2 P24941 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5357681 0.75 CASP1 (0.41) CYP11B2ARGRIA1CACNG8CASP1
SCHEMBL6468361 0.74 CYP2A6 (0.42) CYP11B2ARCDK4CDK2
SCHEMBL3076212 0.73 IKBKB (0.49) CYP11B2TRPV4NSD2ARCYP11B1
SCHEMBL5365964 0.73 CYP11B2 (0.47) CYP11B2TRPV4ARCYP11B1MAOA
SCHEMBL24186806 0.71 CYP11B2 (0.44) CYP11B2TRPV4NSD2ARCYP11B1
SCHEMBL5711187 0.70 CYP11B2 (0.54) CYP11B2TRPV4ARCYP11B1GRIA1
SCHEMBL6890109 0.68 AR (0.53) NSD2AR
SCHEMBL18666733 0.67 CYP11B2 (0.50) CYP11B2TRPV4NSD2ARCYP11B1
SCHEMBL410587 0.66 TRPV4 (0.57) CYP11B2TRPV4ARMAOAMAOB
SCHEMBL11560121 0.66 CYP11B2 (0.49) CYP11B2TRPV4NSD2ARCYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed