SCHEMBL5365964

SCHEMBL5365964

Cc1cc(-c2ccc(C#N)c(Cl)c2)c(C)[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 4/20 0.47
KDM4E B2RXH2 3/20 0.43
HPGD P15428 3/20 0.43
ALDH1A1 P00352 2/20 0.43
GALR3 O60755 1/20 0.43
GAA P10253 1/20 0.43
TRPV4 Q9HBA0 1/20 0.42
PDE3B Q13370 2/20 0.41
PDE3A Q14432 2/20 0.41
PDE5A O76074 1/20 0.41
LMNA P02545 1/20 0.41
TSHR P16473 1/20 0.41
PTGS1 P23219 1/20 0.41
PDE4A P27815 1/20 0.41
CYP2C19 P33261 1/20 0.41
BLM P54132 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
SLC22A12 Q96S37 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5364904 0.78 AR (0.62) AR
SCHEMBL6196775 0.76 ESR2 (0.46) TSHRAR
SCHEMBL4921058 0.75 ALDH1A1 (0.45) CYP11B2KDM4EHPGDALDH1A1GALR3
SCHEMBL11560121 0.74 CYP11B2 (0.49) CYP11B2TRPV4SLC22A12CYP11B1AR
SCHEMBL5358282 0.73 CYP11B2 (0.41) CYP11B2TRPV4CYP11B1ARMAOA
SCHEMBL2320354 0.72 AHR (0.41) KDM4EHPGDGAAPDE3BPDE3A
SCHEMBL5357681 0.72 CASP1 (0.41) CYP11B2KDM4EHPGDALDH1A1GALR3
SCHEMBL9205179 0.71 CYP11B2 (0.52) CYP11B2TRPV4SLC22A12CYP11B1AR
SCHEMBL24186806 0.70 CYP11B2 (0.44) CYP11B2HPGDALDH1A1TRPV4CYP11B1
SCHEMBL6197205 0.70 KCNH2 (0.44) KDM4EALDH1A1PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed