SCHEMBL5358296

SCHEMBL5358296

FC(F)(F)c1cc(CBr)nn1COCc1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.36
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
GAA P10253 1/20 0.35
HPGD P15428 1/20 0.35
HTR2C P28335 4/20 0.34
SLC6A4 P31645 4/20 0.34
HTR2A P28223 1/20 0.34
TACR1 P25103 4/20 0.34
MAPT P10636 1/20 0.33
APP P05067 1/20 0.33
GRN P28799 1/20 0.33
SORT1 Q99523 1/20 0.33
SLC16A3 O15427 1/20 0.32
PDE2A O00408 1/20 0.32
BRD4 O60885 1/20 0.32
POLB P06746 1/20 0.32
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32
CACNA1F O60840 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5367786 0.76 TSHR (0.39) TSHRALDH1A1KDM4EGAAHPGD
SCHEMBL3900724 0.70 PTGS1 (0.43) ALDH1A1KDM4EHPGDMAPTPOLB
SCHEMBL19584627 0.69 NR1H2 (0.44) TSHRKDM4EGAAHPGDHTR2C
SCHEMBL5363641 0.67 TSHR (0.40) TSHRALDH1A1KDM4EHTR2CSLC6A4
SCHEMBL15701583 0.64 PTGS2 (0.45) KDM4EGAAHPGDGRNSORT1
SCHEMBL5464352 0.64 TSHR (0.40) TSHRALDH1A1HTR2CSLC6A4HTR2A
SCHEMBL8157722 0.62 ALDH1A1 (0.61) TSHRALDH1A1KDM4ETACR1POLB
SCHEMBL2226540 0.62 SLC16A3 (0.56) ALDH1A1KDM4EGAAMAPTGRN
Bromoethane SCHEMBL20577437 0.62 TSHR (0.75) TSHRALDH1A1KDM4ETACR1MAPT
SCHEMBL14061138 0.61 SMN1; SMN2 (0.46) TSHRALDH1A1KDM4EGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed