SCHEMBL5360039

SCHEMBL5360039

Nc1nc(N)c2cc(I)ccc2n1

nearest known ligand 0.66

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
DCPS Q96C86 1/20 0.53
DHFR P00374 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21500701 0.81 HTT (0.64)
SCHEMBL29767521 0.81 APP (0.42) DHFR
SCHEMBL30376225 0.81 HTT (0.64)
Quinazoline-2,4,6-Triamine SCHEMBL335027 0.79 DCPS (0.57) DCPSDHFR
Quinazoline-2,4,6-Triamine SCHEMBL30050079 0.79 DCPS (0.57) DCPSDHFR
SCHEMBL27556561 0.77 CYP1A1 (0.69)
SCHEMBL4358438 0.76 HTT (0.68) DCPSDHFR
SCHEMBL29649743 0.76 HTT (0.68) DCPSDHFR
SCHEMBL4755412 0.76 DCPS (0.53) DCPSDHFR
SCHEMBL6679745 0.76 HRH4 (0.58) DCPSDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7256197-B2 Methods for synthesis of diarylmethanes DANA-FARBER CANCER INSTITUTE (US) 2007-08-14 US disclosed
US-20040267011-A1 Methods for synthesis of diarylmethanes DANA-FARBER CANCER INSTITUTE 2004-12-30 US disclosed
US-20040092515-A1 Diaminoquinazoline esters for use as dihydrofolate reductase inhibitors MELACURE THERAPEUTICS AB (SE) 2004-05-13 US disclosed
EP-1366028-A1 DIAMINOQUINAZOLINE ESTERS FOR USE AS DIHYDROFOLATE REDUCTASE INHIBITORS Melacure Therapeutics AB (SE) 2003-12-03 EP disclosed
WO-2003031458-A1 METHODS FOR SYNTHESIS OF DIARYLMETHANES DANA-FARBER CANCER INSTITUTE (US) 2003-04-17 WO disclosed
WO-2002068397-A1 DIAMINOQUINAZOLINE ESTERS FOR USE AS DIHYDROFOLATE REDUCTADE INHIBITORS MELACURE THERAPEUTICS AB (SE) 2002-09-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040092515-A1 Diaminoquinazoline esters for use as dihydrofolate reductase inhibitors DHFR, DPYD, DHODH DCPS 671/4885DHFR 1/4885
US-20040267011-A1 Methods for synthesis of diarylmethanes DHFR, DPYD, DHODH DCPS 778/4885DHFR 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.