SCHEMBL21500701

SCHEMBL21500701

Nc1nc(Cl)nc2ccc(I)cc12

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.64
CYP1A1 P04798 2/20 0.40
CYP1A2 P05177 2/20 0.40
CYP1B1 Q16678 2/20 0.40
TYMS P04818 1/20 0.40
APP P05067 1/20 0.39
HTR3A P46098 1/20 0.38
HRH4 Q9H3N8 1/20 0.38
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30376225 1.00 HTT (0.64) HTTCYP1A1CYP1A2CYP1B1TYMS
SCHEMBL29441517 0.81 HTT (0.68) HTTHTR3AHRH4ALDH1A1
SCHEMBL21500731 0.81 HTT (0.68) HTTHTR3AHRH4ALDH1A1
SCHEMBL1069650 0.81 HTT (0.41) HTTTYMSAPPKDM4EALDH1A1
SCHEMBL5360039 0.81 DCPS (0.53)
SCHEMBL8897424 0.78 HTT (1.00) HTTCYP1A2
SCHEMBL8900878 0.78 HTT (0.64) HTTTYMS
SCHEMBL29767521 0.78 APP (0.42) HTTCYP1A1CYP1A2CYP1B1TYMS
SCHEMBL1069686 0.78 HTT (0.39) HTTTYMSAPPKDM4EALDH1A1
SCHEMBL3778992 0.78 HTT (0.64) HTTHTR3AHRH4KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210353626-A1 BETA-ADRENERGIC RECEPTOR ALLOSTERIC MODULATORS Friedrich-Alexander-Universität Erlangen-Nürnberg (DE) 2021-11-18 US disclosed
WO-2019204768-A1 BETA-ADRENERGIC RECEPTOR ALLOSTERIC MODULATORS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-10-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210353626-A1 BETA-ADRENERGIC RECEPTOR ALLOSTERIC MODULATORS ADRB1, ADRB2, ADRA2B HTT 4394/4885CYP1A1 2625/4885CYP1A2 2202/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.