SCHEMBL5360159

SCHEMBL5360159

CC[Si](CC)(CC)OC(C1CCC(N(CC(F)(F)F)S(=O)(=O)Cc2ccccc2)CC1)(C(F)(F)F)C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RORC P51449 16/20 0.40
USP2 O75604 1/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
ESR2 Q92731 1/20 0.34
CNR2 P34972 1/20 0.32
HSP90AA1 P07900 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1460750 0.79 RORC (0.50) RORCUSP2HPGDHSD17B10ESR2
SCHEMBL5352146 0.78 DRD2 (0.43) RORCUSP2HPGDHSD17B10
SCHEMBL5357408 0.72 SLC6A2 (0.39)
SCHEMBL5348999 0.71 ACHE (0.44)
SCHEMBL5347919 0.71 ACHE (0.44)
SCHEMBL5354218 0.71 HTR1A (0.44)
SCHEMBL13434175 0.68 HSD17B10 (0.54) RORCUSP2HPGDHSD17B10CNR2
SCHEMBL5359018 0.64
SCHEMBL1459811 0.63 ESR2 (0.58) RORCESR2
SCHEMBL7608221 0.63 USP2 (0.50) RORCUSP2HPGDHSD17B10CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1831158-A1 NOVEL CYCLOHEXANE DERIVATIVES F. Hoffmann-Roche AG (CH) 2007-09-12 EP disclosed
US-7253282-B2 Hexafluoroisopropanol substituted cyclohexane derivatives HOFFMAN-LA ROCHE INC. (US) 2007-08-07 US disclosed
WO-2006066779-A1 NOVEL CYCLOHEXANE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2006-06-29 WO disclosed
US-20060135601-A1 Novel hexafluoroisopropanol substituted cyclohexane derivatives HOFFMANN-LA ROCHE INC. 2006-06-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060135601-A1 Novel hexafluoroisopropanol substituted cyclohexane derivatives NR1H3, NR1H2, NR1I2 RORC 161/4885USP2 3697/4885HPGD 2559/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.