SCHEMBL5360267

SCHEMBL5360267

O=C(NC(CCc1ccccc1)C1(O)CCNCC1)c1ccc(O)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.48
MEN1 O00255 2/20 0.48
HTT P42858 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
HPGD P15428 1/20 0.45
HSP90AA1 P07900 1/20 0.44
DPP4 P27487 2/20 0.43
CTSG P08311 3/20 0.41
CTRB1 P17538 3/20 0.41
ADRB2 P07550 1/20 0.40
PRSS1 P07477 2/20 0.39
CMA1 P23946 2/20 0.39
LMNA P02545 1/20 0.39
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39
GRIN2B Q13224 2/20 0.39
HDAC1 Q13547 1/20 0.38
ERAP1 Q9NZ08 2/20 0.38
LNPEP Q9UIQ6 2/20 0.38
ERAP2 Q6P179 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5360592 0.93 KMT2A (0.43) KMT2AMEN1HTTSMN1; SMN2HPGD
SCHEMBL5374718 0.88 RAB9A (0.41) KMT2AMEN1HTTSMN1; SMN2CTRB1
SCHEMBL5363936 0.87 KMT2A (0.44) KMT2AMEN1HTTSMN1; SMN2HPGD
SCHEMBL5368445 0.81 KMT2A (0.40) KMT2AMEN1HTTSMN1; SMN2HPGD
SCHEMBL5370680 0.72 KMT2A (0.44) KMT2AMEN1HTTSMN1; SMN2HPGD
SCHEMBL5363812 0.71 KMT2A (0.46) KMT2AMEN1HTTSMN1; SMN2HPGD
SCHEMBL5362924 0.70 KMT2A (0.41) KMT2AMEN1HTTSMN1; SMN2HPGD
SCHEMBL2472052 0.69 CTRB1 (0.46) HPGDCTRB1HDAC1
SCHEMBL5371067 0.68 NPC1 (0.42) SMN1; SMN2CTRB1
SCHEMBL5375114 0.68 KMT2A (0.42) KMT2AMEN1HTTSMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed