SCHEMBL5360585

SCHEMBL5360585

Cc1c(C#N)c(-c2cccc(C#N)c2)c(C)n1Cc1cc(C(F)(F)F)n[nH]1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AR P10275 6/20 0.42
SYK P43405 2/20 0.37
ALPL P05186 1/20 0.36
ALPI P09923 1/20 0.36
MAP4K4 O95819 1/20 0.36
GSK3A P49840 1/20 0.36
MAT2A P31153 1/20 0.36
ADORA2A P29274 1/20 0.35
ADORA2B P29275 1/20 0.35
ADORA1 P30542 1/20 0.35
SDHB P21912 1/20 0.35
GRIN1 Q05586 2/20 0.34
GRIN2B Q13224 2/20 0.34
PIK3R1 P27986 1/20 0.34
PIK3CA P42336 1/20 0.34
IDO1 P14902 1/20 0.34
GRM2 Q14416 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5359725 0.74 AR (0.48) ARSDHB
SCHEMBL5357164 0.74 CYP11B2 (0.39) ARSDHBPIK3R1PIK3CA
SCHEMBL5366156 0.71 AR (0.37) ARSDHB
SCHEMBL5357454 0.71 AR (0.36) AR
SCHEMBL6468892 0.71 AR (0.77) ARGRIN1GRIN2B
SCHEMBL4262482 0.71 IDO1 (0.49) SYKALPLALPIMAP4K4GSK3A
SCHEMBL5353540 0.71 CYP11B2 (0.38) ARSDHB
SCHEMBL5361524 0.70 AR (0.54) AR
SCHEMBL5362074 0.70 CYP11B2 (0.35) ARSDHB
SCHEMBL6466379 0.69 AR (0.76) AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed