SCHEMBL536178

SCHEMBL536178

CCC1CCCCN1c1ccc(C(=O)OC(=O)c2ccc(-c3ccccc3C)c(CN(C)C)c2)cc1COC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 6/20 0.39
NR1I2 O75469 1/20 0.34
SMARCA2 P51531 1/20 0.34
SMARCA4 P51532 1/20 0.34
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34
PBRM1 Q86U86 1/20 0.34
ALDH1A1 P00352 2/20 0.34
TSHR P16473 2/20 0.34
ALOX15 P16050 1/20 0.34
PLA2G7 Q13093 1/20 0.34
MAPT P10636 3/20 0.34
HTT P42858 1/20 0.34
HIF1A Q16665 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
S1PR3 Q99500 2/20 0.32
FFAR1 O14842 2/20 0.32
KDM4E B2RXH2 3/20 0.32
AR P10275 1/20 0.32
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL536177 0.93 S1PR1 (0.39) S1PR1NR1I2SMARCA2SMARCA4NR1H2
SCHEMBL3466223 0.79 S1PR1 (0.37) S1PR1NR1I2SMARCA2SMARCA4NR1H2
SCHEMBL406995 0.77 S1PR1 (0.49) S1PR1ALDH1A1TSHRALOX15MAPT
SCHEMBL536674 0.76 S1PR1 (0.39) S1PR1NR1I2SMARCA2SMARCA4NR1H2
SCHEMBL536095 0.72 BRD4 (0.35) NR1I2SMARCA2SMARCA4NR1H2PBRM1
SCHEMBL410449 0.71 MEN1 (0.45) S1PR1ALDH1A1TSHRMAPTL3MBTL1
SCHEMBL409947 0.68 S1PR1 (0.52) S1PR1NR1I2SMARCA2SMARCA4NR1H2
SCHEMBL319975 0.68 S1PR1 (0.46) S1PR1ALDH1A1TSHRMAPTL3MBTL1
SCHEMBL409177 0.65 ALDH1A1 (0.51) S1PR1ALDH1A1LMNA
SCHEMBL408083 0.65 GFER (0.46) S1PR1L3MBTL1KDM4EGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414342-A1 OXADIAZOLE DERIVATIVES Merck Serono S.A. (CH) 2012-02-08 EP disclosed
WO-2010112461-A1 OXADIAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2010-10-07 WO disclosed