SCHEMBL536177

SCHEMBL536177

CCC1CCCCN1c1ccc(C(=O)O)cc1COC.Cc1ccccc1-c1ccc(C(=O)O)cc1CN(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 6/20 0.39
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
HIF1A Q16665 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
NR1I2 O75469 1/20 0.35
SMARCA2 P51531 1/20 0.35
SMARCA4 P51532 1/20 0.35
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
PBRM1 Q86U86 1/20 0.35
S1PR3 Q99500 2/20 0.34
PLA2G7 Q13093 1/20 0.34
TSHR P16473 2/20 0.34
POLB P06746 1/20 0.34
FFAR1 O14842 3/20 0.34
DRD2 P14416 1/20 0.33
DRD4 P21917 1/20 0.33
HRH2 P25021 1/20 0.33
HRH1 P35367 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL536178 0.93 S1PR1 (0.39) S1PR1MAPTHTTHIF1AL3MBTL1
SCHEMBL3466223 0.86 S1PR1 (0.37) S1PR1MAPTHTTHIF1AL3MBTL1
SCHEMBL406995 0.85 S1PR1 (0.49) S1PR1MAPTHTTHIF1AL3MBTL1
SCHEMBL536674 0.84 S1PR1 (0.39) S1PR1MAPTHIF1AL3MBTL1NR1I2
SCHEMBL409177 0.75 ALDH1A1 (0.51) S1PR1POLB
SCHEMBL319590 0.74 S1PR1 (0.52) S1PR1S1PR3POLBFFAR1
SCHEMBL2482448 0.73 S1PR1 (0.35) S1PR1NR3C2
SCHEMBL408083 0.73 GFER (0.46) S1PR1L3MBTL1POLBNR3C2HPGD
SCHEMBL536094 0.71 PRKG1 (0.38) HTTNR1I2SMARCA2SMARCA4NR1H2
SCHEMBL410352 0.70 GFER (0.42) L3MBTL1POLBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414342-A1 OXADIAZOLE DERIVATIVES Merck Serono S.A. (CH) 2012-02-08 EP disclosed
WO-2010112461-A1 OXADIAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2010-10-07 WO disclosed