SCHEMBL5362174

SCHEMBL5362174

Cc1c(-c2ccc(C#N)cc2)c(C(F)(F)F)c(C)n1Cc1cn(C(c2ccccc2)(c2ccccc2)c2ccccc2)nn1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AR P10275 8/20 0.44
CYP19A1 P11511 5/20 0.35
PIN1 Q13526 1/20 0.33
TACR1 P25103 1/20 0.33
KIF11 P52732 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6525379 0.88 AR (0.58) ARCYP19A1PIN1
SCHEMBL5358210 0.87 AR (0.47) ARCYP19A1PIN1
SCHEMBL14347623 0.75 AR (0.42) ARKIF11
SCHEMBL5358573 0.74 AR (0.54) ARKIF11
SCHEMBL5369671 0.73 AR (0.60) AR
SCHEMBL5365095 0.71 AR (0.65) ARCYP19A1
SCHEMBL6466386 0.71 AR (0.58) ARCYP19A1
SCHEMBL6466161 0.65 AR (0.58) AR
SCHEMBL5359676 0.64 AR (0.53) AR
SCHEMBL5364107 0.64 AR (0.56) ARCYP19A1TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed