SCHEMBL5358210

SCHEMBL5358210

Cc1c(I)c(-c2ccc(C#N)cc2)c(C)n1Cc1cn(C(c2ccccc2)(c2ccccc2)c2ccccc2)nn1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AR P10275 7/20 0.47
CYP19A1 P11511 9/20 0.37
PIN1 Q13526 1/20 0.35
BAZ2B Q9UIF8 1/20 0.33
BAZ2A Q9UIF9 1/20 0.33
ACSS2 Q9NR19 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6525379 0.91 AR (0.58) ARCYP19A1PIN1BAZ2BBAZ2A
SCHEMBL5362174 0.87 AR (0.44) ARCYP19A1PIN1
SCHEMBL5369671 0.76 AR (0.60) ARACSS2
SCHEMBL6466386 0.73 AR (0.58) ARCYP19A1BAZ2BBAZ2A
SCHEMBL5365095 0.73 AR (0.65) ARCYP19A1
SCHEMBL5358573 0.70 AR (0.54) AR
SCHEMBL6466161 0.67 AR (0.58) ARACSS2
SCHEMBL5359676 0.66 AR (0.53) AR
SCHEMBL6464955 0.66 NOTUM (0.36) CYP19A1
SCHEMBL3852265 0.65 KIF11 (0.37) CYP19A1BAZ2BBAZ2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed