SCHEMBL5362471

SCHEMBL5362471

NC(=O)COc1ccc(S(=O)(=O)Cl)cc1OCC(N)=O

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.48
PTGDR2 Q9Y5Y4 1/20 0.42
SNCA P37840 1/20 0.42
HTT P42858 2/20 0.41
KDM4E B2RXH2 1/20 0.41
KMT2A Q03164 2/20 0.41
LMNA P02545 3/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
GAA P10253 1/20 0.38
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5366352 0.85 PTGDR2 (0.50) ALDH1A1PTGDR2SMN1; SMN2CYP2C19
SCHEMBL5359690 0.85 ALDH1A1 (0.49) ALDH1A1PTGDR2SNCAHTTKDM4E
SCHEMBL5367144 0.78 ALDH1A1 (0.51) ALDH1A1KDM4EKMT2ALMNAGAA
SCHEMBL2564265 0.76 ALDH1A1 (0.47) ALDH1A1HTTKMT2ALMNASMN1; SMN2
SCHEMBL9092236 0.76 ALDH1A1 (0.53) ALDH1A1KDM4EKMT2ASMN1; SMN2CYP2C19
SCHEMBL4808533 0.74 PTGDR2 (0.51) PTGDR2
SCHEMBL6165389 0.73 TDP1 (0.64) PTGDR2HTTSMN1; SMN2CYP2C19GAA
SCHEMBL5761411 0.72 ALDH1A1 (0.38) ALDH1A1PTGDR2HTTKDM4EKMT2A
SCHEMBL8322727 0.72 ALDH1A1 (0.59) ALDH1A1HTTKDM4EKMT2ALMNA
SCHEMBL5363756 0.72 LMNA (0.62) ALDH1A1HTTKMT2ALMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7294716-B2 Process for preparing isomerically pure prodrugs of proton pump inhibitors ALLERGAN, INC. (US) 2007-11-13 US disclosed
US-7294716-B2 Process for preparing isomerically pure prodrugs of proton pump inhibitors ALLERGAN, INC. (US) 2007-11-13 US disclosed
US-7294716-B2 Process for preparing isomerically pure prodrugs of proton pump inhibitors ALLERGAN, INC. (US) 2007-11-13 US disclosed
EP-1644352-A1 PROCESS FOR PREPARING ISOMERICALLY PURE PRODRUGS OF PROTON PUMP INHIBITORS Allergan, Inc. (US) 2006-04-12 EP disclosed
WO-2005016917-A1 PROCESS FOR PREPARING ISOMERICALLY PURE PRODRUGS OF PROTON PUMP INHIBITORS ALLERGAN, INC. (US) 2005-02-24 WO disclosed
US-20050038076-A1 Process for preparing isomerically pure prodrugs of proton pump inhibitors ALEVIUM PHARMACEUTICALS, INC. 2005-02-17 US disclosed
US-6559167-B1 Prodrugs of the pyridyl methyl sulfinyl benzimidazole type proton pump inhibitor drugs have a hydrolyzable arylsulfonyl or heteroarylsulfonyl group attached to the benzimidazole nitrogen. The prodrugs of the invention hydrolyze under REGENTS OF THE UNIVERSITY OF CALIFORNIA 2003-05-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050038076-A1 Process for preparing isomerically pure prodrugs of proton pump inhibitors SI, ATP6AP1, HRH2 ALDH1A1 1650/4885PTGDR2 484/4885SNCA 3558/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.